← Mechanisms of action
CHRM3
SINGLE PROTEINHomo sapiens
Preferred name: Muscarinic acetylcholine receptor M3 ChEMBL ↗
Linked proteins
Drugs acting on this target (54)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| asp8302 | Activator | experimental | Small molecule | CHRM3 activator |
| acetylcholine chloride (miochol) | Agonist | approved | Small molecule | CHRM3 agonist |
| bethanechol (urecholine) | Agonist | approved | Small molecule | CHRM3 agonist |
| carbachol (miostat) | Agonist | approved | Small molecule | CHRM3 agonist |
| cevimeline hydrochloride (evoxac) | Agonist | approved | Small molecule | CHRM3 agonist |
| methacholine (provocholine) | Agonist | approved | Small molecule | CHRM3 agonist |
| pilocarpine (ocusert) | Agonist | approved | Small molecule | CHRM3 agonist |
| aclidinium (tudorza pressair) | Antagonist | approved | Small molecule | CHRM3 antagonist |
| anisotropine methylbromide (valpin) | Antagonist | approved | Small molecule | CHRM3 antagonist |
| asm-024 | Antagonist | experimental | Small molecule | CHRM3 antagonist |
| atropine | Antagonist | approved | Small molecule | CHRM3 antagonist |
| azd-9164 | Antagonist | experimental | Small molecule | Muscarinic acetylcholine receptor M3 antagonist |
| azd8683 | Antagonist | experimental | Small molecule | CHRM3 antagonist |
| batefenterol | Antagonist | experimental | Small molecule | CHRM3 antagonist |
| chf6366 | Antagonist | experimental | Small molecule | CHRM3 antagonist |
| clidinium (quarzan) | Antagonist | approved | Small molecule | CHRM3 antagonist |
| cyclopentolate (cyclogyl) | Antagonist | approved | Small molecule | CHRM3 antagonist |
| cyclopropylmethylscopolamine | Antagonist | experimental | Small molecule | CHRM3 antagonist |
| da-8010 | Antagonist | experimental | Small molecule | CHRM3 antagonist |
| darifenacin (enablex) | Antagonist | approved | Small molecule | CHRM3 antagonist |
| dicyclomine hydrochloride (bentyl) | Antagonist | approved | Small molecule | CHRM3 antagonist |
| diphemanil methylsulfate (prantal) | Antagonist | approved | Small molecule | CHRM3 antagonist |
| fesoterodine (toviaz) | Antagonist | approved | Small molecule | CHRM3 antagonist |
| glycopyrronium (robinul) | Antagonist | approved | Small molecule | CHRM3 antagonist |
| hexocyclium methylsulfate (tral) | Antagonist | approved | Small molecule | CHRM3 antagonist |
| imidafenacin | Antagonist | experimental | Small molecule | Muscarinic acetylcholine receptor M3 antagonist |
| ipratropium (atrovent) | Antagonist | approved | Small molecule | CHRM3 antagonist |
| isopropamide iodide (darbid) | Antagonist | approved | Small molecule | CHRM3 antagonist |
| las-190792 | Antagonist | experimental | Small molecule | CHRM3 antagonist |
| mepenzolate bromide (cantil) | Antagonist | approved | Small molecule | CHRM3 antagonist |
| methylscopolamine bromide | Antagonist | approved | Small molecule | CHRM3 antagonist |
| oxitropium (Oxivent) | Antagonist | experimental | Small molecule | CHRM3 antagonist |
| oxybutynin (ditropan) | Antagonist | approved | Small molecule | CHRM3 antagonist |
| oxyphencyclimine (daricon) | Antagonist | approved | Small molecule | CHRM3 antagonist |
| oxyphenonium (antrenyl) | Antagonist | approved | Small molecule | CHRM3 antagonist |
| penehyclidine | Antagonist | experimental | Small molecule | CHRM3 antagonist |
| propantheline bromide (pro-banthine) | Antagonist | approved | Small molecule | CHRM3 antagonist |
| qax028 | Antagonist | experimental | Small molecule | CHRM3 antagonist |
| revefenacin (yupelri) | Antagonist | approved | Small molecule | Muscarinic acetylcholine receptor M3 antagonist |
| sofpironium (SOFDRA) | Antagonist | approved | Small molecule | CHRM3 antagonist |
| solifenacin (vesicare) | Antagonist | approved | Small molecule | CHRM3 antagonist |
| tarafenacin | Antagonist | experimental | Small molecule | CHRM3 antagonist |
| tiotropium (spiriva) | Antagonist | approved | Small molecule | CHRM3 antagonist |
| tolterodine (detrol) | Antagonist | approved | Small molecule | CHRM3 antagonist |
| tridihexethyl | Antagonist | approved | Small molecule | CHRM3 antagonist |
| tropicamide (mydriacyl) | Antagonist | approved | Small molecule | CHRM3 antagonist |
| trospium (sanctura) | Antagonist | approved | Small molecule | CHRM3 antagonist |
| umeclidinium (incruse ellipta) | Antagonist | approved | Small molecule | CHRM3 antagonist |
| aroxybutynin | Inhibitor | experimental | Small molecule | CHRM3 inhibitor |
| gantacurium | Inhibitor | experimental | Small molecule | GPM3 inhibitor |
| nifekalant | Inhibitor | experimental | Small molecule | CHRM3 inhibitor |
| r-oxybutynin | Inhibitor | experimental | Small molecule | CHRM3 inhibitor |
| v0162 | Inhibitor | experimental | Small molecule | CHRM3 inhibitor |
| talsaclidine | Partial agonist | experimental | Small molecule | Muscarinic acetylcholine receptor M3 partial agonist |