← Mechanisms of action
Muscarinic acetylcholine receptor
PROTEIN FAMILYHomo sapiens
Linked proteins
Drugs acting on this target (12)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| aceclidine (Vizz) | Agonist | approved | Small molecule | Muscarinic acetylcholine receptor agonist |
| afacifenacin | Antagonist | experimental | Small molecule | Muscarinic acetylcholine receptor antagonist |
| darotropium | Antagonist | experimental | Small molecule | Muscarinic acetylcholine receptor antagonist |
| glycopyrronium (robinul) | Antagonist | approved | Small molecule | Muscarinic acetylcholine receptor antagonist |
| hyoscyamine | Antagonist | experimental | Small molecule | Muscarinic acetylcholine receptor antagonist |
| Laventair | Antagonist | experimental | Small molecule | Muscarinic acetylcholine receptor antagonist |
| revefenacin (yupelri) | Antagonist | approved | Small molecule | Muscarinic acetylcholine receptor antagonist |
| terodiline | Antagonist | experimental | Small molecule | Muscarinic acetylcholine receptor antagonist |
| tiropramide | Antagonist | experimental | Small molecule | Muscarinic acetylcholine receptor antagonist |
| glycopyrronium (robinul) | Inhibitor | approved | Small molecule | Muscarinic acetylcholine receptor inhibitor |
| mebeverine | Inhibitor | experimental | Small molecule | Muscarinic acetylcholine receptor inhibitor |
| sofpironium (SOFDRA) | Inhibitor | approved | Small molecule | Muscarinic acetylcholine receptor inhibitor |