← Mechanisms of action
DRD2
SINGLE PROTEINHomo sapiens
Preferred name: Dopamine D2 receptor ChEMBL ↗
Linked proteins
Drugs acting on this target (90)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| cabergoline (dostinex) | Agonist | approved | Small molecule | DRD2 agonist |
| d390 | Agonist | experimental | Small molecule | DRD2 agonist |
| lu ae04621 | Agonist | experimental | Small molecule | DRD2 agonist |
| lu af28996 | Agonist | experimental | Small molecule | DRD2 agonist |
| lu ag06479 | Agonist | experimental | Small molecule | DRD2 agonist |
| pf-00217830 | Agonist | experimental | Small molecule | DRD2 agonist |
| phno | Agonist | experimental | Small molecule | DRD2 agonist |
| Piribedil | Agonist | experimental | Small molecule | DRD2 agonist |
| quinagolide (Norprolac) | Agonist | experimental | Small molecule | DRD2 agonist |
| sumanirole | Agonist | experimental | Small molecule | DRD2 agonist |
| tbr-760 | Agonist | experimental | Small molecule | DRD2 agonist |
| ac-201 | Antagonist | experimental | Small molecule | DRD2 antagonist |
| acetophenazine (tindal) | Antagonist | approved | Small molecule | DRD2 antagonist |
| alizapride | Antagonist | experimental | Small molecule | DRD2 antagonist |
| asenapine (saphris) | Antagonist | approved | Small molecule | DRD2 antagonist |
| ati-9242 | Antagonist | experimental | Small molecule | DRD2 antagonist |
| Benperidol (glianimon) | Antagonist | experimental | Small molecule | DRD2 antagonist |
| blonanserin (Lonasen) | Antagonist | experimental | Small molecule | Dopamine D2 receptor antagonist |
| bromperidol (tesoprel) | Antagonist | experimental | Small molecule | DRD2 antagonist |
| carphenazine (proketazine) | Antagonist | approved | Small molecule | DRD2 antagonist |
| chlorprothixene (taractan) | Antagonist | approved | Small molecule | DRD2 antagonist |
| clebopride maleate | Antagonist | experimental | Small molecule | DRD2 antagonist |
| clozapine (clozaril) | Antagonist | approved | Small molecule | DRD2 antagonist |
| cvl-936 | Antagonist | experimental | Small molecule | DRD2 antagonist |
| Deudomperidone | Antagonist | experimental | Small molecule | DRD2 antagonist |
| domperidone | Antagonist | experimental | Small molecule | DRD2 antagonist |
| enx-104 | Antagonist | experimental | Small molecule | DRD2 antagonist |
| enx-205 | Antagonist | experimental | Small molecule | DRD2 antagonist |
| fluphenazine (permitil) | Antagonist | approved | Small molecule | DRD2 antagonist |
| iloperidone (fanapt) | Antagonist | approved | Small molecule | DRD2 antagonist |
| itropride | Antagonist | experimental | Small molecule | Dopamine D2 receptor antagonist |
| jnj-37822681 | Antagonist | experimental | Small molecule | DRD2 antagonist |
| levosulpiride | Antagonist | experimental | Small molecule | Dopamine D2 receptor antagonist |
| lurasidone (latuda) | Antagonist | approved | Small molecule | DRD2 antagonist |
| Menatetrenone (MK-4) | Antagonist | experimental | Small molecule | DRD2 antagonist |
| mesoridazine (serentil) | Antagonist | approved | Small molecule | DRD2 antagonist |
| metoclopramide (reglan) | Antagonist | approved | Small molecule | DRD2 antagonist |
| metopimazine | Antagonist | experimental | Small molecule | DRD2 antagonist |
| molindone (moban) | Antagonist | approved | Small molecule | DRD2 antagonist |
| onc206 | Antagonist | experimental | Small molecule | DRD2 antagonist |
| paliperidone (invega) | Antagonist | approved | Small molecule | DRD2 antagonist |
| perphenazine (trilafon) | Antagonist | approved | Small molecule | DRD2 antagonist |
| piperacetazine (quide) | Antagonist | approved | Small molecule | Dopamine D2 receptor antagonist |
| prochlorperazine (compazine) | Antagonist | approved | Small molecule | DRD2 antagonist |
| quetiapine (seroquel) | Antagonist | approved | Small molecule | DRD2 antagonist |
| raclopride | Antagonist | experimental | Small molecule | DRD2 antagonist |
| remoxipride | Antagonist | experimental | Small molecule | DRD2 antagonist |
| risperidone (risperdal) | Antagonist | approved | Small molecule | DRD2 antagonist |
| sb773812 | Antagonist | experimental | Small molecule | DRD2 antagonist |
| sertindole (Serdolect) | Antagonist | experimental | Small molecule | DRD2 antagonist |
| sulpiride | Antagonist | experimental | Small molecule | Dopamine D2 receptor antagonist |
| thiethylperazine (torecan) | Antagonist | approved | Small molecule | DRD2 antagonist |
| thiothixene (navane) | Antagonist | approved | Small molecule | DRD2 antagonist |
| tiaprizal | Antagonist | experimental | Small molecule | Dopamine D2 receptor antagonist |
| triflupromazine (vesprin) | Antagonist | approved | Small molecule | DRD2 antagonist |
| trimipramine (surmontil) | Antagonist | approved | Small molecule | DRD2 antagonist |
| veralipride | Antagonist | experimental | Small molecule | DRD2 antagonist |
| ziprasidone (geodon) | Antagonist | approved | Small molecule | DRD2 antagonist |
| zotepine | Antagonist | experimental | Small molecule | DRD2 antagonist |
| zuclopenthixol | Antagonist | experimental | Small molecule | DRD2 antagonist |
| blonanserin (Lonasen) | Inhibitor | experimental | Small molecule | DRD2 inhibitor |
| dordaviprone (Modeyso) | Inhibitor | approved | Small molecule | DRD2 inhibitor |
| fallypride | Inhibitor | experimental | Small molecule | DRD2 inhibitor |
| fluspirilene | Inhibitor | experimental | Small molecule | DRD2 inhibitor |
| gsk1322888 | Inhibitor | experimental | Small molecule | DRD2 inhibitor |
| hec113995pa | Inhibitor | experimental | Small molecule | DRD2 inhibitor |
| levosulpiride | Inhibitor | experimental | Small molecule | DRD2 inhibitor |
| mknd-201 | Inhibitor | experimental | Small molecule | DRD2 inhibitor |
| prothipendyl | Inhibitor | experimental | Small molecule | DRD2 inhibitor |
| tak-906 | Inhibitor | experimental | Small molecule | DRD2 inhibitor |
| tiaprizal | Inhibitor | experimental | Small molecule | DRD2 inhibitor |
| zicronapine | Inhibitor | experimental | Small molecule | DRD2 inhibitor |
| abbv-932 | Modulator | experimental | Small molecule | DRD2 modulator |
| acr325 | Modulator | experimental | Small molecule | DRD2 modulator |
| benzquinamide (emete-con) | Modulator | approved | Small molecule | DRD2 modulator |
| cariprazine (vraylar) | Modulator | approved | Small molecule | DRD2 modulator |
| pridopidine | Modulator | experimental | Small molecule | DRD2 modulator |
| seridopidine | Modulator | experimental | Small molecule | DRD2 modulator |
| trimethobenzamide (tigan) | Other | approved | Small molecule | DRD2 other |
| aripiprazole (abilify) | Partial agonist | approved | Small molecule | DRD2 partial agonist |
| bifeprunoxum | Partial agonist | experimental | Small molecule | DRD2 partial agonist |
| brexpiprazole (rexulti) | Partial agonist | approved | Small molecule | DRD2 partial agonist |
| Brilaroxazine | Partial agonist | experimental | Small molecule | DRD2 partial agonist |
| iti-1284 | Partial agonist | experimental | Small molecule | DRD2 partial agonist |
| lumateperone (Caplyta) | Partial agonist | approved | Small molecule | DRD2 partial agonist |
| osu 6162 | Partial agonist | experimental | Small molecule | DRD2 partial agonist |
| palindore | Partial agonist | experimental | Small molecule | DRD2 partial agonist |
| pf-00217830 | Partial agonist | experimental | Small molecule | Dopamine D2 receptor partial agonist |
| sarizotan | Partial agonist | experimental | Small molecule | DRD2 partial agonist |
| xc130-a10h | Partial agonist | experimental | Small molecule | DRD2 partial agonist |