← Mechanisms of action
CHRM1
SINGLE PROTEINHomo sapiens
Preferred name: Muscarinic acetylcholine receptor M1 ChEMBL ↗
Linked proteins
Drugs acting on this target (56)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| acp-104 | Activator | experimental | Small molecule | CHRM1 activator |
| Desmethylclozapine | Activator | experimental | Small molecule | CHRM1 activator |
| mk-7622 | Activator | experimental | Small molecule | CHRM1 activator |
| tak-071 | Activator | experimental | Small molecule | CHRM1 activator |
| vu319 | Activator | experimental | Small molecule | CHRM1 activator |
| acetyl-ß-methylcholine | Agonist | experimental | Small molecule | CHRM1 agonist |
| cevimeline hydrochloride (evoxac) | Agonist | approved | Small molecule | CHRM1 agonist |
| htl0009936 | Agonist | experimental | Small molecule | CHRM1 agonist |
| minaprine | Agonist | experimental | Small molecule | CHRM1 agonist |
| ml-007c-ma | Agonist | experimental | Small molecule | CHRM1 agonist |
| ngx267 | Agonist | experimental | Small molecule | CHRM1 agonist |
| pilocarpine (ocusert) | Agonist | approved | Small molecule | CHRM1 agonist |
| talsaclidine | Agonist | experimental | Small molecule | Muscarinic acetylcholine receptor M1 agonist |
| xanomeline (Cobenfy) | Agonist | approved | Small molecule | Muscarinic acetylcholine receptor M1 agonist |
| anisodine | Antagonist | experimental | Small molecule | CHRM1 antagonist |
| anisotropine methylbromide (valpin) | Antagonist | approved | Small molecule | CHRM1 antagonist |
| asm-024 | Antagonist | experimental | Small molecule | CHRM1 antagonist |
| atropine | Antagonist | approved | Small molecule | CHRM1 antagonist |
| azd9164 | Antagonist | experimental | Small molecule | CHRM1 antagonist |
| benzatropine (cogentin) | Antagonist | approved | Small molecule | CHRM1 antagonist |
| biperiden (akineton) | Antagonist | approved | Small molecule | CHRM1 antagonist |
| clidinium (quarzan) | Antagonist | approved | Small molecule | CHRM1 antagonist |
| cycrimine (pagitane) | Antagonist | approved | Small molecule | CHRM1 antagonist |
| dicyclomine hydrochloride (bentyl) | Antagonist | approved | Small molecule | CHRM1 antagonist |
| diphemanil methylsulfate (prantal) | Antagonist | approved | Small molecule | CHRM1 antagonist |
| diphenidol (vontrol) | Antagonist | approved | Small molecule | CHRM1 antagonist |
| ethopropazine (parsidol) | Antagonist | approved | Small molecule | CHRM1 antagonist |
| glycopyrronium (robinul) | Antagonist | approved | Small molecule | CHRM1 antagonist |
| hexocyclium methylsulfate (tral) | Antagonist | approved | Small molecule | CHRM1 antagonist |
| imidafenacin | Antagonist | experimental | Small molecule | Muscarinic acetylcholine receptor M1 antagonist |
| isopropamide iodide (darbid) | Antagonist | approved | Small molecule | CHRM1 antagonist |
| mepenzolate bromide (cantil) | Antagonist | approved | Small molecule | CHRM1 antagonist |
| methylscopolamine bromide | Antagonist | approved | Small molecule | CHRM1 antagonist |
| metixene (trest) | Antagonist | approved | Small molecule | CHRM1 antagonist |
| oxyphencyclimine (daricon) | Antagonist | approved | Small molecule | CHRM1 antagonist |
| oxyphenonium (antrenyl) | Antagonist | approved | Small molecule | CHRM1 antagonist |
| penehyclidine | Antagonist | experimental | Small molecule | CHRM1 antagonist |
| procyclidine hydrochloride (kemadrin) | Antagonist | approved | Small molecule | CHRM1 antagonist |
| propantheline bromide (pro-banthine) | Antagonist | approved | Small molecule | CHRM1 antagonist |
| qax028 | Antagonist | experimental | Small molecule | CHRM1 antagonist |
| scopolamine (transderm scop) | Antagonist | approved | Small molecule | CHRM1 antagonist |
| telenzepine | Antagonist | experimental | Small molecule | CHRM1 antagonist |
| tridihexethyl | Antagonist | approved | Small molecule | CHRM1 antagonist |
| trihexyphenidyl | Antagonist | approved | Small molecule | CHRM1 antagonist |
| Acotiamide | Inhibitor | experimental | Small molecule | CHRM1 inhibitor |
| anavex3-71 | Inhibitor | experimental | Small molecule | CHRM1 inhibitor |
| aroxybutynin | Inhibitor | experimental | Small molecule | CHRM1 inhibitor |
| nbi-1117570 | Inhibitor | experimental | Small molecule | CHRM1 inhibitor |
| pipe-307 | Inhibitor | experimental | Small molecule | CHRM1 inhibitor |
| pirenzepine | Inhibitor | experimental | Small molecule | CHRM1 inhibitor |
| r-oxybutynin | Inhibitor | experimental | Small molecule | CHRM1 inhibitor |
| azd6088 | Partial agonist | experimental | Small molecule | CHRM1 partial agonist |
| htl0018318 | Partial agonist | experimental | Small molecule | CHRM1 partial agonist |
| mk-7622 | Positive allosteric modulator | experimental | Small molecule | Muscarinic acetylcholine receptor M1 positive allosteric modulator |
| suvn-i6107 | Positive allosteric modulator | experimental | Small molecule | CHRM1 positive allosteric modulator |
| tak-071 | Positive allosteric modulator | experimental | Small molecule | Muscarinic acetylcholine receptor M1 positive allosteric modulator |