← Mechanisms of action
Epidermal growth factor receptor
PROTEIN FAMILYHomo sapiens
Linked proteins
Drugs acting on this target (40)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| epidermal growth factor | Agonist | experimental | Recombinant protein | Epidermal growth factor receptor agonist |
| amivantamab-vmjw (Rybrevant) | Antagonist | approved | mAb | Epidermal growth factor receptor antagonist |
| icotinib (Conmana) | Antagonist | experimental | Small molecule | Epidermal growth factor receptor antagonist |
| mobocertinib (EXKIVITY) | Antagonist | approved | Small molecule | Epidermal growth factor receptor antagonist |
| ty-9591 | Antagonist | experimental | Small molecule | Epidermal growth factor receptor antagonist |
| cart-egfr-il13ra2 | Binding agent | experimental | Cell therapy | Epidermal growth factor receptor binding agent |
| Losatuxizumab vedotin | Binding agent | experimental | mAb | Epidermal growth factor receptor binding agent |
| egf vaccine | Immunity, active | experimental | Vaccine | Epidermal growth factor receptor immunity, active |
| pep-3 vaccine | Immunity, active | experimental | Vaccine | Epidermal growth factor receptor immunity, active |
| abivertinib | Inhibitor | experimental | Small molecule | Epidermal growth factor receptor inhibitor |
| ac0010ma | Inhibitor | experimental | Small molecule | Epidermal growth factor receptor inhibitor |
| almonertinib | Inhibitor | experimental | Small molecule | Epidermal growth factor receptor inhibitor |
| asp-1929 | Inhibitor | experimental | Small molecule | Epidermal growth factor receptor inhibitor |
| aumolertinib | Inhibitor | experimental | Small molecule | Epidermal growth factor receptor inhibitor |
| Befotertinib | Inhibitor | experimental | Small molecule | Epidermal growth factor receptor inhibitor |
| bibw 2948 bs | Inhibitor | experimental | Small molecule | Epidermal growth factor receptor inhibitor |
| bpi-361175 | Inhibitor | experimental | Small molecule | Epidermal growth factor receptor inhibitor |
| dacomitinib (vizimpro) | Inhibitor | approved | Small molecule | Epidermal growth factor receptor inhibitor |
| egfrviii peptide | Inhibitor | experimental | Peptide | Epidermal growth factor receptor inhibitor |
| erlotinib (tarceva) | Inhibitor | approved | Small molecule | Epidermal growth factor receptor inhibitor |
| furmonertinib (Ives) | Inhibitor | experimental | Small molecule | Epidermal growth factor receptor inhibitor |
| hemay020 | Inhibitor | experimental | Small molecule | Epidermal growth factor receptor inhibitor |
| hki-357 | Inhibitor | experimental | Small molecule | Epidermal growth factor receptor inhibitor |
| Larotinib | Inhibitor | experimental | Small molecule | Epidermal growth factor receptor inhibitor |
| lazertinib (Lazcluze) | Inhibitor | approved | Small molecule | Epidermal growth factor receptor inhibitor |
| limertinib | Inhibitor | experimental | Small molecule | Epidermal growth factor receptor inhibitor |
| naquotinib | Inhibitor | experimental | Small molecule | Epidermal growth factor receptor inhibitor |
| nazartinib | Inhibitor | experimental | Small molecule | Epidermal growth factor receptor inhibitor |
| neratinib maleate (nerlynx) | Inhibitor | approved | Small molecule | Epidermal growth factor receptor inhibitor |
| nituzumab | Inhibitor | experimental | mAb | Epidermal growth factor receptor inhibitor |
| Oritinib | Inhibitor | experimental | Small molecule | Epidermal growth factor receptor inhibitor |
| osimertinib (tagrisso) | Inhibitor | approved | Small molecule | Epidermal growth factor receptor inhibitor |
| pf-06459988 | Inhibitor | experimental | Small molecule | Epidermal growth factor receptor inhibitor |
| poziotinib | Inhibitor | experimental | Small molecule | Epidermal growth factor receptor inhibitor |
| Rezivertinib | Inhibitor | experimental | Small molecule | Epidermal growth factor receptor inhibitor |
| sklb1028 | Inhibitor | experimental | Small molecule | Epidermal growth factor receptor inhibitor |
| sunvozertinib (Zegfrovy) | Inhibitor | approved | Small molecule | Epidermal growth factor receptor inhibitor |
| tarloxotinib | Inhibitor | experimental | Small molecule | Epidermal growth factor receptor inhibitor |
| vandetanib (caprelsa) | Inhibitor | approved | Small molecule | Epidermal growth factor receptor inhibitor |
| zn-e4 | Inhibitor | experimental | Small molecule | Epidermal growth factor receptor inhibitor |