← Mechanisms of action

ERBB4

SINGLE PROTEINHomo sapiens
Preferred name: Receptor protein-tyrosine kinase erbB-4 ChEMBL ↗

Linked proteins

Drugs acting on this target (12)

Active Pharmaceutical Ingredient Mechanism Type Approval Status API Type Mechanism of Action
afatinib (gilotrif)InhibitorapprovedSmall moleculeERBB4 inhibitor
bms-599626InhibitorexperimentalSmall moleculeERBB4 inhibitor
bms-690514InhibitorexperimentalSmall moleculeERBB4 inhibitor
canertinibInhibitorexperimentalSmall moleculeERBB4 inhibitor
dacomitinib (vizimpro)InhibitorapprovedSmall moleculeERBB4 inhibitor
fcn-411InhibitorexperimentalSmall moleculeERBB4 inhibitor
jnj-26483327InhibitorexperimentalSmall moleculeERBB4 inhibitor
neratinib maleate (nerlynx)InhibitorapprovedSmall moleculeReceptor protein-tyrosine kinase erbB-4 inhibitor
pirotinibInhibitorexperimentalSmall moleculeERBB4 inhibitor
pyrrolitinibInhibitorexperimentalSmall moleculeERBB4 inhibitor
tarloxotinibInhibitorexperimentalSmall moleculeERBB4 inhibitor
tas2940InhibitorexperimentalSmall moleculeERBB4 inhibitor