Rezivertinib

Small moleculeexperimental

Clinical trial activity

5 trials · 3 clinical orgs · 0 marketing orgs

Phase 1
3
Phase 2
2
Phase 3
1
Phase 4
0

Earliest trial started Aug 16, 2017 (NCT03386955)

Timeline

2010s

  1. Jan 1, 2017

    Earliest Phase 1 Sponsor(trial)

  2. Jan 1, 2019

    Earliest Phase 2 Sponsor(trial)

  3. Jan 1, 2019

    Earliest Phase 3 Sponsor(trial)

Indications

Mechanism of action

Chemistry & pharmacology

Loading structure…

SMILES

C=CC(=O)Nc1cc(Nc2nccc(-c3cn(C)c4ccccc34)n2)c(OC)cc1OCCN(C)C
Mol. weight
486.58 g/mol
Lipinski Ro5
Pass
Rule of 3
No
Chirality
Achiral Molecule
Inorganic
No
Polymer
No

Oral

No

Parenteral

No

Topical

No

Sources

Clinical trials

NCT IDPhaseStart dateSponsor(s)
NCT04135820Phase 1Nov 30, 2019Beta Pharma, Inc., Jiao Tong University
NCT04135833Phase 1Nov 30, 2019Beta Pharma, Inc., Jiao Tong University
NCT03866499Phase 3May 31, 2019Beta Pharma, Inc., Chinese Academy of Medical Sciences
NCT03812809Phase 2Apr 1, 2019Beta Pharma, Inc., Chinese Academy of Medical Sciences
NCT03386955Phase 1Aug 16, 2017Beta Pharma, Inc., Chinese Academy of Medical Sciences
Showing 5 of 5 trials
Page 1 / 1

Organizations

Research & Development (3)

OrganizationOrg typeTrialsAs lead sponsorPhasesEarliest year
Beta Pharma, Inc.For profit5532017
Chinese Academy of Medical SciencesAcademic/Hospital3032017
Jiao Tong UniversityAcademic/Hospital2012019
3 organizations
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