← Mechanisms of action
Cyclooxygenase
PROTEIN FAMILYHomo sapiens
Linked proteins
Drugs acting on this target (60)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| mefenamic acid (ponstel) | Antagonist | approved | Small molecule | Cyclooxygenase antagonist |
| acetaminophen (tylenol) | Inhibitor | approved | Small molecule | Cyclooxygenase inhibitor |
| acetylsalicylic acid (aspirin) | Inhibitor | approved | Small molecule | Cyclooxygenase inhibitor |
| aliviador | Inhibitor | experimental | Small molecule | Cyclooxygenase inhibitor |
| aminophenazone cyclamate | Inhibitor | experimental | Small molecule | Cyclooxygenase inhibitor |
| aminosalicylic acid (Paser) | Inhibitor | approved | Small molecule | Cyclooxygenase inhibitor |
| azapropazone | Inhibitor | experimental | Small molecule | Cyclooxygenase inhibitor |
| balsalazide (colazal) | Inhibitor | approved | Small molecule | Cyclooxygenase inhibitor |
| benzydamine | Inhibitor | experimental | Small molecule | Cyclooxygenase inhibitor |
| bismuth subsalicylate (Pepto-Bismol) | Inhibitor | approved | Small molecule | Cyclooxygenase inhibitor |
| bromfenac (xibrom) | Inhibitor | approved | Small molecule | Cyclooxygenase inhibitor |
| Carbasalate | Inhibitor | experimental | Small molecule | Cyclooxygenase inhibitor |
| clometacin | Inhibitor | experimental | Small molecule | Cyclooxygenase inhibitor |
| Dexketoprofen | Inhibitor | experimental | Small molecule | Cyclooxygenase inhibitor |
| diclofenac (voltaren) | Inhibitor | approved | Small molecule | Cyclooxygenase inhibitor |
| diethylamine salicylate | Inhibitor | experimental | Small molecule | Cyclooxygenase inhibitor |
| diflunisal (dolobid) | Inhibitor | approved | Small molecule | Cyclooxygenase inhibitor |
| esflurbiprofen | Inhibitor | experimental | Small molecule | Cyclooxygenase inhibitor |
| fenclofenac | Inhibitor | experimental | Small molecule | Cyclooxygenase inhibitor |
| fenoprofen (nalfon) | Inhibitor | approved | Small molecule | Cyclooxygenase inhibitor |
| flufenamic acid | Inhibitor | experimental | Small molecule | Cyclooxygenase inhibitor |
| flurbiprofen (ansaid) | Inhibitor | approved | Small molecule | Cyclooxygenase inhibitor |
| gingerol | Inhibitor | experimental | Small molecule | Cyclooxygenase inhibitor |
| glafenine | Inhibitor | experimental | Small molecule | Cyclooxygenase inhibitor |
| ibufenac | Inhibitor | experimental | Small molecule | Cyclooxygenase inhibitor |
| ibuprofen (motrin) | Inhibitor | approved | Small molecule | Cyclooxygenase inhibitor |
| idea-070 | Inhibitor | experimental | Small molecule | Cyclooxygenase inhibitor |
| indobufen | Inhibitor | experimental | Small molecule | Cyclooxygenase inhibitor |
| indomethacin (indocin) | Inhibitor | approved | Small molecule | Cyclooxygenase inhibitor |
| indoprofen | Inhibitor | experimental | Small molecule | Cyclooxygenase inhibitor |
| isoxicam | Inhibitor | experimental | Small molecule | Cyclooxygenase inhibitor |
| jnj-10450232 | Inhibitor | experimental | Small molecule | Cyclooxygenase inhibitor |
| ketoprofen (orudis) | Inhibitor | approved | Small molecule | Cyclooxygenase inhibitor |
| ketorolac (acuvail) | Inhibitor | approved | Small molecule | Cyclooxygenase inhibitor |
| lobenzarit | Inhibitor | experimental | Small molecule | Cyclooxygenase inhibitor |
| lornoxicam | Inhibitor | experimental | Small molecule | Cyclooxygenase inhibitor |
| loxoprofen | Inhibitor | experimental | Small molecule | Cyclooxygenase inhibitor |
| meclofenamic acid (meclomen) | Inhibitor | approved | Small molecule | Cyclooxygenase inhibitor |
| mefenamic acid (ponstel) | Inhibitor | approved | Small molecule | Cyclooxygenase inhibitor |
| metamizole (Novalgin) | Inhibitor | experimental | Small molecule | Cyclooxygenase inhibitor |
| naproxen (naprosyn) | Inhibitor | approved | Small molecule | Cyclooxygenase inhibitor |
| nepafenac (nevanac) | Inhibitor | approved | Small molecule | Cyclooxygenase inhibitor |
| nitroaspirin | Inhibitor | experimental | Small molecule | Cyclooxygenase inhibitor |
| olsalazine (dipentum) | Inhibitor | approved | Small molecule | Cyclooxygenase inhibitor |
| oxaprozin (daypro) | Inhibitor | approved | Small molecule | Cyclooxygenase inhibitor |
| oxyphenbutazone (Tandearil) | Inhibitor | approved | Small molecule | Cyclooxygenase inhibitor |
| p3914 | Inhibitor | experimental | Small molecule | Cyclooxygenase inhibitor |
| phenylbutazone (butazolidin) | Inhibitor | approved | Small molecule | Cyclooxygenase inhibitor |
| piroxicam (feldene) | Inhibitor | approved | Small molecule | Cyclooxygenase inhibitor |
| pirprofen | Inhibitor | experimental | Small molecule | Cyclooxygenase inhibitor |
| rantudil | Inhibitor | experimental | Small molecule | Cyclooxygenase inhibitor |
| salicylic acid | Inhibitor | marketed | Small molecule | Cyclooxygenase inhibitor |
| sulfasalazine (azulfidine) | Inhibitor | approved | Small molecule | Cyclooxygenase inhibitor |
| sulindac (clinoril) | Inhibitor | approved | Small molecule | Cyclooxygenase inhibitor |
| suprofen (Profenal) | Inhibitor | withdrawn | Small molecule | Cyclooxygenase inhibitor |
| tenoxicam | Inhibitor | experimental | Small molecule | Cyclooxygenase inhibitor |
| tinoridine | Inhibitor | experimental | Small molecule | Cyclooxygenase inhibitor |
| tolmetin (tolectin) | Inhibitor | approved | Small molecule | Cyclooxygenase inhibitor |
| triflusal | Inhibitor | experimental | Small molecule | Cyclooxygenase inhibitor |
| dihomo-gamma-linolenic acid | Substrate | experimental | Small molecule | Cyclooxygenase substrate |