← Mechanisms of action
ADRB2
SINGLE PROTEINHomo sapiens
Preferred name: Beta-2 adrenergic receptor ChEMBL ↗
Linked proteins
Drugs acting on this target (62)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| Etafedrine | Activator | experimental | Small molecule | ADRB2 activator |
| abediterol | Agonist | experimental | Small molecule | ADRB2 agonist |
| albuterol (proventil) | Agonist | approved | Small molecule | ADRB2 agonist |
| ar08 | Agonist | experimental | Small molecule | ADRB2 agonist |
| arformoterol (brovana) | Agonist | approved | Small molecule | ADRB2 agonist |
| atr-258 | Agonist | experimental | Small molecule | ADRB2 agonist |
| azd-3199 | Agonist | experimental | Small molecule | ADRB2 agonist |
| bambuterol | Agonist | experimental | Small molecule | Beta-2 adrenergic receptor agonist |
| batefenterol | Agonist | experimental | Small molecule | ADRB2 agonist |
| bedoradrine | Agonist | experimental | Small molecule | ADRB2 agonist |
| bitolterol (tornalate) | Agonist | approved | Small molecule | ADRB2 agonist |
| clenbuterol | Agonist | experimental | Small molecule | ADRB2 agonist |
| cst-2032 | Agonist | experimental | Small molecule | ADRB2 agonist |
| dbm-1152a | Agonist | experimental | Small molecule | ADRB2 agonist |
| dilevalol | Agonist | experimental | Small molecule | ADRB2 agonist |
| dobutamine (dobutrex) | Agonist | approved | Small molecule | ADRB2 agonist |
| fenoterol | Agonist | experimental | Small molecule | ADRB2 agonist |
| formoterol (foradil) | Agonist | approved | Small molecule | ADRB2 agonist |
| gsk159797 | Agonist | experimental | Small molecule | ADRB2 agonist |
| gsk159802 | Agonist | experimental | Small molecule | ADRB2 agonist |
| indacaterol (arcapta neohaler) | Agonist | approved | Small molecule | ADRB2 agonist |
| indicaterol | Agonist | experimental | Small molecule | ADRB2 agonist |
| isoetharine (bronkosol) | Agonist | approved | Small molecule | ADRB2 agonist |
| isoxsuprine | Agonist | experimental | Small molecule | ADRB2 agonist |
| las-190792 | Agonist | experimental | Small molecule | ADRB2 agonist |
| levalbuterol (xopenex) | Agonist | approved | Small molecule | ADRB2 agonist |
| metaproterenol (alupent) | Agonist | approved | Small molecule | ADRB2 agonist |
| olodaterol (striverdi respimat) | Agonist | approved | Small molecule | ADRB2 agonist |
| pf-00610355 | Agonist | experimental | Small molecule | Beta-2 adrenergic receptor agonist |
| pirbuterol (maxair) | Agonist | approved | Small molecule | ADRB2 agonist |
| procaterol | Agonist | experimental | Small molecule | ADRB2 agonist |
| protokylol (ventaire) | Agonist | approved | Small molecule | ADRB2 agonist |
| reproterol | Agonist | experimental | Small molecule | ADRB2 agonist |
| rimoterol | Agonist | experimental | Small molecule | Beta-2 adrenergic receptor agonist |
| ritodrine (yutopar) | Agonist | approved | Small molecule | ADRB2 agonist |
| salmeterol (serevent) | Agonist | approved | Small molecule | ADRB2 agonist |
| ta-2005 | Agonist | experimental | Small molecule | ADRB2 agonist |
| terbutaline (bricanyl) | Agonist | approved | Small molecule | ADRB2 agonist |
| tulobuterol | Agonist | experimental | Small molecule | Beta-2 adrenergic receptor agonist |
| vilanterol (Anoro Elipta) | Agonist | approved | Small molecule | ADRB2 agonist |
| bucindolol | Antagonist | experimental | Small molecule | Beta-2 adrenergic receptor antagonist |
| esmolol (brevibloc) | Antagonist | approved | Small molecule | ADRB2 antagonist |
| levobunolol (betagan) | Antagonist | approved | Small molecule | ADRB2 antagonist |
| ly-377604 | Antagonist | experimental | Small molecule | ADRB2 antagonist |
| metipranolol (optipranolol) | Antagonist | approved | Small molecule | ADRB2 antagonist |
| nadolol (corgard) | Antagonist | approved | Small molecule | ADRB2 antagonist |
| nebivolol (bystolic) | Antagonist | approved | Small molecule | ADRB2 antagonist |
| oxprenolol (trasicor) | Antagonist | approved | Small molecule | ADRB2 antagonist |
| penbutolol (levatol) | Antagonist | approved | Small molecule | ADRB2 antagonist |
| pronetalol | Antagonist | experimental | Small molecule | ADRB2 antagonist |
| propafenone (rythmol) | Antagonist | approved | Small molecule | ADRB2 antagonist |
| propanolol | Antagonist | experimental | Small molecule | ADRB2 antagonist |
| propranolol (inderal) | Antagonist | approved | Small molecule | ADRB2 antagonist |
| sotalol (betapace) | Antagonist | approved | Small molecule | ADRB2 antagonist |
| timolol (blocadren) | Antagonist | approved | Small molecule | ADRB2 antagonist |
| tulobuterol | Antagonist | experimental | Small molecule | ADRB2 antagonist |
| syl040012 | Antisense inhibitor | experimental | Nucleic acid | ADRB2 antisense inhibitor |
| centhaquine | Inhibitor | experimental | Small molecule | ADRB2 inhibitor |
| ci 775 | Inhibitor | experimental | Small molecule | ADRB2 inhibitor |
| tr4 | Inhibitor | experimental | Small molecule | ADRB2 inhibitor |
| celiprolol | Partial agonist | experimental | Small molecule | ADRB2 partial agonist |
| pindolol (visken) | Partial agonist | approved | Small molecule | ADRB2 partial agonist |