← Mechanisms of action
Estrogen receptor
PROTEIN FAMILYHomo sapiens
Linked proteins
Drugs acting on this target (54)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| conjugated equine estrogens (Premarin) | Agonist | approved | Animal product | Estrogen receptor agonist |
| conjugated estrogen | Agonist | experimental | Animal product | Estrogen receptor agonist |
| diethylstilbestrol diphosphate (stilphostrol) | Agonist | withdrawn | Small molecule | Estrogen receptor agonist |
| estetrol (NEXTSTELLIS) | Agonist | approved | Small molecule | Estrogen receptor agonist |
| estriol | Agonist | experimental | Small molecule | Estrogen receptor agonist |
| estrogen | Agonist | experimental | Animal product | Estrogen receptor agonist |
| gsk232802 | Agonist | experimental | Small molecule | Estrogen receptor agonist |
| lasofoxifene | Agonist | experimental | Small molecule | Estrogen receptor agonist |
| mk-6913 | Agonist | experimental | Small molecule | Estrogen receptor agonist |
| orageston | Agonist | experimental | Small molecule | Estrogen receptor agonist |
| promestriene | Agonist | experimental | Small molecule | Estrogen receptor agonist |
| quinestrol (estrovis) | Agonist | approved | Small molecule | Estrogen receptor agonist |
| ttc-352 | Agonist | experimental | Small molecule | Estrogen receptor agonist |
| fulvestrant (faslodex) | Antagonist | approved | Small molecule | Estrogen receptor antagonist |
| Giredestrant | Antagonist | experimental | Small molecule | Estrogen receptor antagonist |
| lx-039 | Antagonist | experimental | Small molecule | Estrogen receptor antagonist |
| op-1250 | Antagonist | experimental | Small molecule | Estrogen receptor antagonist |
| tqb3915 | Antagonist | experimental | Small molecule | estrogen receptor |
| ac682 | Degrader | experimental | Small molecule | Estrogen receptor degrader |
| ac699 | Degrader | experimental | Small molecule | estrogen receptor |
| and019 | Degrader | experimental | Small molecule | Estrogen receptor degrader |
| dalpiciclib | Degrader | experimental | Small molecule | Estrogen receptor degrader |
| fwd1802 | Degrader | experimental | Small molecule | Estrogen receptor degrader |
| hrs-1358 | Degrader | experimental | Small molecule | Estrogen receptor degrader |
| sco-120 | Degrader | experimental | Small molecule | Estrogen receptor degrader |
| scr-6852 | Degrader | experimental | Small molecule | Estrogen receptor |
| acolbifene | Inhibitor | experimental | Small molecule | Estrogen receptor inhibitor |
| azd9496 | Inhibitor | experimental | Small molecule | Estrogen receptor inhibitor |
| d-0502 | Inhibitor | experimental | Small molecule | Estrogen receptor inhibitor |
| g1t48 | Inhibitor | experimental | Small molecule | Estrogen receptor inhibitor |
| gdc-0810 | Inhibitor | experimental | Small molecule | Estrogen receptor inhibitor |
| sar439859 | Inhibitor | experimental | Small molecule | Estrogen receptor inhibitor |
| zb716 | Inhibitor | experimental | Small molecule | Estrogen receptor inhibitor |
| zn-c5 | Inhibitor | experimental | Small molecule | Estrogen receptor inhibitor |
| afimoxifene | Modulator | experimental | Small molecule | Estrogen receptor modulator |
| arzoxifene | Modulator | experimental | Small molecule | Estrogen receptor modulator |
| bazedoxifene (Duavee) | Modulator | approved | Small molecule | Estrogen receptor modulator |
| cc-8490 | Modulator | experimental | Small molecule | Estrogen receptor modulator |
| chf-4227 | Modulator | experimental | Small molecule | Estrogen receptor modulator |
| custirsen | Modulator | experimental | Nucleic acid | Estrogen receptor modulator |
| cyclofenil | Modulator | experimental | Small molecule | Estrogen receptor modulator |
| droloxifene | Modulator | experimental | Small molecule | Estrogen receptor modulator |
| enclomiphene | Modulator | experimental | Small molecule | Estrogen receptor modulator |
| estriol | Modulator | experimental | Small molecule | Estrogen receptor modulator |
| fispemifene | Modulator | experimental | Small molecule | Estrogen receptor modulator |
| idoxifene | Modulator | experimental | Small molecule | Estrogen receptor modulator |
| imlunestrant | Modulator | approved | Small molecule | Estrogen receptor modulator |
| lasofoxifene | Modulator | experimental | Small molecule | Estrogen receptor modulator |
| ly2245461 | Modulator | experimental | Small molecule | Estrogen receptor modulator |
| ospemifene (osphena) | Modulator | approved | Small molecule | Estrogen receptor modulator |
| pipendoxifene | Modulator | experimental | Small molecule | Estrogen receptor modulator |
| ritlecitinib (Litfulo) | Modulator | approved | Small molecule | Estrogen receptor modulator |
| toremifene (fareston) | Modulator | approved | Small molecule | Estrogen receptor modulator |
| trans-clomiphene | Modulator | experimental | Small molecule | Estrogen receptor modulator |