idoxifene
Small moleculeexperimental
Clinical trial activity
0 trials · 0 clinical orgs · 0 marketing orgs
Phase 1
0
Phase 2
0
Phase 3
0
Phase 4
0
Mechanism of action
- Estrogen receptorMODULATOR
Estrogen receptor modulator
SERM, development stopped as ineffective compared to tamoxifen.
Chemistry & pharmacology
Loading structure…
SMILES
CC/C(=C(\c1ccc(I)cc1)c1ccc(OCCN2CCCC2)cc1)c1ccccc1- Mol. weight
- 523.46 g/mol
- Lipinski Ro5
- 2 violation(s)
- Rule of 3
- No
- Chirality
- Achiral Molecule
- Inorganic
- No
- Polymer
- No
Oral
No
Parenteral
No
Topical
No
Sources
- ChEMBLCHEMBL6318 ↗
Also known as
- 1-(4-iodophenyl)-1-(4-(2-pyrrolidinoethoxy)phenyl)-2-phenyl-1-butene
- 4-iodopyrrolidinotamoxifen
- cb-7432
- cb-7432
- idoxifene
- idoxifene
- idoxifene
- pyr-i-tam
- pyrrolidino-4-iodotamoxifen
- sb-223030
- sb-223030