← Mechanisms of action
ESR1
SINGLE PROTEINHomo sapiens
Preferred name: Estrogen receptor alpha ChEMBL ↗
Linked proteins
Drugs acting on this target (29)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| bisphenol a | Activator | experimental | Small molecule | ESR1 activator |
| dienestrol | Agonist | approved | Small molecule | ESR1 agonist |
| diethylstilbestrol (Fosfestrol) | Agonist | approved | Small molecule | ESR1 agonist |
| estradiol (progynon depot) | Agonist | approved | Small molecule | ESR1 agonist |
| estrone | Agonist | approved | Small molecule | ESR1 agonist |
| ethinyl estradiol (Estinyl) | Agonist | approved | Small molecule | ESR1 agonist |
| gtx-758 | Agonist | experimental | Small molecule | ESR1 agonist |
| mestranol | Agonist | approved | Small molecule | ESR1 agonist |
| polyestradiol (Estradurin) | Agonist | approved | Small molecule | ESR1 agonist |
| fulvestrant (faslodex) | Antagonist | approved | Small molecule | Estrogen receptor alpha antagonist |
| h3b-6545 | Antagonist | experimental | Small molecule | ESR1 antagonist |
| ts-108 | Antagonist | experimental | Small molecule | ESR1 antagonist |
| camizestrant | Degrader | experimental | Small molecule | Estrogen receptor alpha degrader |
| elacestrant (Orserdu) | Degrader | approved | Small molecule | ESR1 degrader |
| fulvestrant (faslodex) | Degrader | approved | Small molecule | Estrogen receptor degrader |
| gdc-0927 | Degrader | experimental | Small molecule | ESR1 degrader |
| Giredestrant | Degrader | experimental | Small molecule | Estrogen receptor alpha degrader |
| hp568 | Degrader | experimental | Small molecule | ESR1 degrader |
| sar439859 | Degrader | experimental | Small molecule | Estrogen receptor alpha degrader |
| vepdegestrant | Degrader | experimental | Small molecule | ESR1 degrader |
| dimethandrolone undecanoate | Disrupting agent | experimental | Small molecule | ESR1 disrupting agent |
| erx-315 | Inhibitor | experimental | Small molecule | ESR1 inhibitor |
| indole-3-carbinol | Inhibitor | experimental | Small molecule | ESR1 inhibitor |
| lsz102 | Inhibitor | experimental | Small molecule | ESR1 inhibitor |
| shr9549 | Inhibitor | experimental | Small molecule | ESR1 inhibitor |
| camizestrant | Modulator | experimental | Small molecule | ESR1 modulator |
| clomifene (clomid) | Modulator | approved | Small molecule | ESR1 modulator |
| endoxifen | Modulator | experimental | Small molecule | ESR1 modulator |
| tamoxifen (nolvadex) | Modulator | approved | Small molecule | ESR1 modulator |