← Mechanisms of action

ESR2

SINGLE PROTEINHomo sapiens
Preferred name: Estrogen receptor beta ChEMBL ↗

Linked proteins

Drugs acting on this target (11)

Active Pharmaceutical Ingredient Mechanism Type Approval Status API Type Mechanism of Action
bay 86-5310AgonistexperimentalSmall moleculeESR2 agonist
bio 300AgonistexperimentalSmall moleculeESR2 agonist
cr1447AgonistexperimentalSmall moleculeESR2 agonist
erb-257AgonistexperimentalSmall moleculeESR2 agonist
erteberelAgonistexperimentalSmall moleculeESR2 agonist
mf101AgonistexperimentalSmall moleculeESR2 agonist
prinaberelAgonistexperimentalSmall moleculeESR2 agonist
s-equolAgonistexperimentalSmall moleculeESR2 agonist
vg101InhibitorexperimentalSmall moleculeESR2 inhibitor
chlorotrianisene (tace)ModulatorapprovedSmall moleculeESR2 modulator
estramustine (emcyt)ModulatorapprovedSmall moleculeESR2 modulator