← Mechanisms of action
NR3C1
SINGLE PROTEINHomo sapiens
Preferred name: Glucocorticoid receptor ChEMBL ↗
Linked proteins
Drugs acting on this target (73)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| alclometasone (aclovate) | Agonist | approved | Small molecule | NR3C1 agonist |
| amcinonide (cyclocort) | Agonist | approved | Small molecule | NR3C1 agonist |
| axr-270 | Agonist | experimental | Small molecule | NR3C1 agonist |
| bay1003803 | Agonist | experimental | Small molecule | NR3C1 agonist |
| beclomethasone (vanceril) | Agonist | approved | Small molecule | NR3C1 agonist |
| betamethasone (celestone) | Agonist | approved | Small molecule | NR3C1 agonist |
| budesonide (rhinocort) | Agonist | approved | Small molecule | NR3C1 agonist |
| ciclesonide (alvesco) | Agonist | approved | Small molecule | NR3C1 agonist |
| clobetasol (dermovate) | Agonist | approved | mAb | NR3C1 agonist |
| clocortolone (cloderm) | Agonist | approved | Small molecule | NR3C1 agonist |
| cortivazol | Agonist | experimental | Small molecule | NR3C1 agonist |
| deflazacort (emflaza) | Agonist | approved | Small molecule | NR3C1 agonist |
| desoximetasone (topicort) | Agonist | approved | Small molecule | NR3C1 agonist |
| dexamethasone | Agonist | approved | Small molecule | NR3C1 agonist |
| diflorasone (FLORONE) | Agonist | approved | Small molecule | NR3C1 agonist |
| difluprednate (durezol) | Agonist | approved | Small molecule | NR3C1 agonist |
| eso-101 | Agonist | experimental | Small molecule | NR3C1 agonist |
| flumethasone (locorten) | Agonist | approved | Small molecule | NR3C1 agonist |
| flunisolide (nasalide) | Agonist | approved | Small molecule | NR3C1 agonist |
| fluocinolone acetonide (synalar) | Agonist | approved | Small molecule | NR3C1 agonist |
| fluocinonide (lidex) | Agonist | approved | Small molecule | NR3C1 agonist |
| fluorometholone (fml) | Agonist | approved | Small molecule | NR3C1 agonist |
| fluprednisolone (alphadrol) | Agonist | approved | Small molecule | NR3C1 agonist |
| flurandrenolide (cordran) | Agonist | approved | Small molecule | NR3C1 agonist |
| fluticasone (cutivate) | Agonist | approved | Small molecule | NR3C1 agonist |
| formocortal | Agonist | experimental | Small molecule | NR3C1 agonist |
| gw870086 | Agonist | experimental | Small molecule | NR3C1 agonist |
| halcinonide (halog) | Agonist | approved | Small molecule | NR3C1 agonist |
| halobetasol (ultravate) | Agonist | approved | Small molecule | NR3C1 agonist |
| halometasone | Agonist | experimental | Small molecule | NR3C1 agonist |
| hydrocortamate (magnacort) | Agonist | approved | Small molecule | NR3C1 agonist |
| hydrocortisone (solu-cortef) | Agonist | approved | Small molecule | NR3C1 agonist |
| leo 134310 | Agonist | experimental | Small molecule | NR3C1 agonist |
| loteprednol (lotemax) | Agonist | approved | Small molecule | NR3C1 agonist |
| mapracorat | Agonist | experimental | Small molecule | NR3C1 agonist |
| medrysone (hms) | Agonist | approved | Small molecule | NR3C1 agonist |
| Methoxypregnenolone | Agonist | experimental | Small molecule | NR3C1 agonist |
| methylprednisolone (medrol) | Agonist | approved | Small molecule | NR3C1 agonist |
| mometasone (elocon) | Agonist | approved | Small molecule | NR3C1 agonist |
| paramethasone acetate (haldrone) | Agonist | approved | Small molecule | NR3C1 agonist |
| prednicarbate (dermatop) | Agonist | approved | Small molecule | NR3C1 agonist |
| prednisolone (hydeltra) | Agonist | approved | Small molecule | NR3C1 agonist |
| prednisone (meticorten) | Agonist | approved | Small molecule | NR3C1 agonist |
| rimexolone (vexol) | Agonist | approved | Small molecule | NR3C1 agonist |
| sodium succinate | Agonist | approved | Small molecule | NR3C1 agonist |
| sparc1316 | Agonist | experimental | Small molecule | NR3C1 agonist |
| triamcinolone (kenalog) | Agonist | approved | Small molecule | NR3C1 agonist |
| ulobetasol propionate (Ultravate) | Agonist | approved | Small molecule | NR3C1 agonist |
| urea | Agonist | approved | Small molecule | NR3C1 agonist |
| vamorolone (Agamree) | Agonist | approved | Small molecule | Glucocorticoid receptor agonist |
| bi 653048 | Antagonist | experimental | Small molecule | NR3C1 antagonist |
| cort 108297 | Antagonist | experimental | Small molecule | NR3C1 antagonist |
| cort-125134 | Antagonist | experimental | Small molecule | NR3C1 antagonist |
| cort118335 | Antagonist | experimental | Small molecule | NR3C1 antagonist |
| cort125281 | Antagonist | experimental | Small molecule | NR3C1 antagonist |
| cort125329 | Antagonist | experimental | Small molecule | NR3C1 antagonist |
| cortisone acetate (cortone) | Antagonist | approved | Small molecule | NR3C1 antagonist |
| cyproviron | Antagonist | experimental | Small molecule | NR3C1 antagonist |
| mifepristone (mifeprex) | Antagonist | approved | Small molecule | NR3C1 antagonist |
| org-34517 | Antagonist | experimental | Small molecule | NR3C1 antagonist |
| relacorilant | Antagonist | experimental | Small molecule | Glucocorticoid receptor antagonist |
| azd5423 | Inhibitor | experimental | Small molecule | NR3C1 inhibitor |
| oric-101 | Inhibitor | experimental | Small molecule | NR3C1 inhibitor |
| PT150 | Inhibitor | experimental | Small molecule | NR3C1 inhibitor |
| relacorilant | Inhibitor | experimental | Small molecule | NR3C1 inhibitor |
| abbv-3373 | Modulator | experimental | mAb | Glucocorticoid receptor modulator |
| azd-5423 | Modulator | experimental | Small molecule | Glucocorticoid receptor modulator |
| dagrocorat | Modulator | experimental | Small molecule | NR3C1 modulator |
| Dazucorilant | Modulator | experimental | Small molecule | NR3C1 modulator |
| fosdagrocorat | Modulator | experimental | Small molecule | NR3C1 modulator |
| miricorilant | Modulator | experimental | Small molecule | NR3C1 modulator |
| Mizacorat | Modulator | experimental | Small molecule | NR3C1 modulator |
| Velsecorat | Modulator | experimental | Small molecule | NR3C1 modulator |