← Mechanisms of action
Bacterial penicillin-binding protein
PROTEIN FAMILYBacteria
Linked proteins
- D-alanyl-D-alanine carboxypeptidase DacB (dacB) ↗
- Peptidoglycan D,D-transpeptidase FtsI (ftsI) ↗
- Penicillin-binding protein 1A (mrcA) ↗
- Penicillin-binding protein 1B (mrcB) ↗
- D-alanyl-D-alanine carboxypeptidase DacA (dacA) ↗
- Peptidoglycan D,D-transpeptidase MrdA (mrdA) ↗
- D-alanyl-D-alanine carboxypeptidase DacC (dacC) ↗
Drugs acting on this target (64)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| cefiderocol (Fetroja) | Antagonist | approved | Small molecule | Bacterial penicillin-binding protein antagonist |
| amoxicillin | Inhibitor | approved | Small molecule | Bacterial penicillin-binding protein inhibitor |
| aztreonam (azactam) | Inhibitor | approved | Small molecule | Bacterial penicillin-binding protein inhibitor |
| bacampicillin (spectrobid) | Inhibitor | approved | Small molecule | Bacterial penicillin-binding protein inhibitor |
| carbenicillin (pyopen) | Inhibitor | approved | Small molecule | Bacterial penicillin-binding protein inhibitor |
| cefaclor (ceclor) | Inhibitor | approved | Small molecule | Bacterial penicillin-binding protein inhibitor |
| cefadroxil (duricef) | Inhibitor | approved | Small molecule | Bacterial penicillin-binding protein inhibitor |
| cefalotin | Inhibitor | approved | Small molecule | Bacterial penicillin-binding protein inhibitor |
| cefamandole (mandol) | Inhibitor | approved | Small molecule | Bacterial penicillin-binding protein inhibitor |
| cefapirin (Cefadyl) | Inhibitor | approved | Small molecule | Bacterial penicillin-binding protein inhibitor |
| cefazolin (ancef) | Inhibitor | approved | Small molecule | Bacterial penicillin-binding protein inhibitor |
| cefdinir (omnicef) | Inhibitor | approved | Small molecule | Bacterial penicillin-binding protein inhibitor |
| cefditoren (spectracef) | Inhibitor | approved | Small molecule | Bacterial penicillin-binding protein inhibitor |
| cefepime (maxipeme) | Inhibitor | approved | Small molecule | Bacterial penicillin-binding protein inhibitor |
| cefiderocol (Fetroja) | Inhibitor | approved | Small molecule | Bacterial penicillin-binding protein inhibitor |
| cefixime (suprax) | Inhibitor | approved | Small molecule | Bacterial penicillin-binding protein inhibitor |
| cefmenoxime (cefmax) | Inhibitor | approved | Small molecule | Bacterial penicillin-binding protein inhibitor |
| cefmetazole (zefazone) | Inhibitor | approved | Small molecule | Bacterial penicillin-binding protein inhibitor |
| cefodizime sodium | Inhibitor | experimental | Small molecule | Bacterial penicillin-binding protein inhibitor |
| cefonicid | Inhibitor | approved | Small molecule | Bacterial penicillin-binding protein inhibitor |
| cefoperazone (cefobid) | Inhibitor | approved | Small molecule | Bacterial penicillin-binding protein inhibitor |
| ceforanide (precef) | Inhibitor | approved | Small molecule | Bacterial penicillin-binding protein inhibitor |
| cefotaxime (claforan) | Inhibitor | approved | Small molecule | Bacterial penicillin-binding protein inhibitor |
| cefotetan (cefotan) | Inhibitor | approved | Small molecule | Bacterial penicillin-binding protein inhibitor |
| cefotiam (ceradon) | Inhibitor | approved | Small molecule | Bacterial penicillin-binding protein inhibitor |
| cefoxitin (mefoxin) | Inhibitor | approved | Small molecule | Bacterial penicillin-binding protein inhibitor |
| cefpiramide | Inhibitor | approved | Small molecule | Bacterial penicillin-binding protein inhibitor |
| cefpirome (cefrom) | Inhibitor | experimental | Small molecule | Bacterial penicillin-binding protein inhibitor |
| cefpodoxime (vantin) | Inhibitor | approved | Small molecule | Bacterial penicillin-binding protein inhibitor |
| cefprozil (cefzil) | Inhibitor | approved | Small molecule | Bacterial penicillin-binding protein inhibitor |
| cefradine | Inhibitor | approved | Small molecule | Bacterial penicillin-binding protein inhibitor |
| cefsulodin sodium salt | Inhibitor | experimental | Small molecule | Bacterial penicillin-binding protein inhibitor |
| ceftaroline fosamil (teflaro) | Inhibitor | approved | Small molecule | Bacterial penicillin-binding protein inhibitor |
| ceftazidime (fortaz) | Inhibitor | approved | Small molecule | Bacterial penicillin-binding protein inhibitor |
| ceftibuten (cedax) | Inhibitor | approved | Small molecule | Bacterial penicillin-binding protein inhibitor |
| ceftizoxime (Cefizox) | Inhibitor | approved | Small molecule | Bacterial penicillin-binding protein inhibitor |
| ceftobiprole (Zevtera) | Inhibitor | approved | Small molecule | Bacterial penicillin-binding protein inhibitor |
| ceftolozane (Zerbaxa) | Inhibitor | approved | Small molecule | Bacterial penicillin-binding protein inhibitor |
| ceftriaxone (rocephin) | Inhibitor | approved | Small molecule | Bacterial penicillin-binding protein inhibitor |
| cefuroxime (zinacef) | Inhibitor | approved | Small molecule | Bacterial penicillin-binding protein inhibitor |
| cephalexin (keflex) | Inhibitor | approved | Small molecule | Bacterial penicillin-binding protein inhibitor |
| cephaloglycin (kafocin) | Inhibitor | approved | Small molecule | Bacterial penicillin-binding protein inhibitor |
| cyclacillin (cyclapen-w) | Inhibitor | approved | Small molecule | Bacterial penicillin-binding protein inhibitor |
| doripenem (doribax) | Inhibitor | approved | Small molecule | Bacterial penicillin-binding protein inhibitor |
| ertapenem (invanz) | Inhibitor | approved | Small molecule | Bacterial penicillin-binding protein inhibitor |
| faropenem medoxomil (Fropenem) | Inhibitor | experimental | Small molecule | Bacterial penicillin-binding protein inhibitor |
| flomoxef (Flumarin) | Inhibitor | experimental | Small molecule | Bacterial penicillin-binding protein inhibitor |
| flucloxacillin | Inhibitor | experimental | Small molecule | Bacterial penicillin-binding protein inhibitor |
| imipenem (primaxin) | Inhibitor | approved | Small molecule | Bacterial penicillin-binding protein inhibitor |
| loracarbef (lorabid) | Inhibitor | approved | Small molecule | Bacterial penicillin-binding protein inhibitor |
| meropenem (merrem) | Inhibitor | approved | Small molecule | Bacterial penicillin-binding protein inhibitor |
| mezlocillin (mezlin) | Inhibitor | approved | Small molecule | Bacterial penicillin-binding protein inhibitor |
| moxalactam (moxam) | Inhibitor | approved | Small molecule | Bacterial penicillin-binding protein inhibitor |
| penamecillin | Inhibitor | experimental | Small molecule | Bacterial penicillin-binding protein inhibitor |
| phenoxymethylpenicillin | Inhibitor | approved | Small molecule | Bacterial penicillin-binding protein inhibitor |
| piperacillin (pipracil) | Inhibitor | approved | Small molecule | Bacterial penicillin-binding protein inhibitor |
| pivampicillin | Inhibitor | experimental | Small molecule | Bacterial penicillin-binding protein inhibitor |
| procaine benzylpenicillin (novocaine) | Inhibitor | approved | Small molecule | Bacterial penicillin-binding protein inhibitor |
| razupenem | Inhibitor | experimental | Small molecule | Bacterial penicillin-binding protein inhibitor |
| sulopenem etzadroxil (Orlynvah) | Inhibitor | approved | Small molecule | Bacterial penicillin-binding protein inhibitor |
| talampicillin hydrochloride | Inhibitor | experimental | Small molecule | Bacterial penicillin-binding protein inhibitor |
| tebipenem | Inhibitor | experimental | Small molecule | Bacterial penicillin-binding protein inhibitor |
| temocillin | Inhibitor | experimental | Small molecule | Bacterial penicillin-binding protein inhibitor |
| ticarcillin (ticar) | Inhibitor | approved | Small molecule | Bacterial penicillin-binding protein inhibitor |