← Mechanisms of action
Adrenergic receptor alpha
PROTEIN FAMILYHomo sapiens
Linked proteins
Drugs acting on this target (14)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| ephedrine | Agonist | approved | Small molecule | Adrenergic receptor alpha agonist |
| epinephrine (levophed) | Agonist | approved | Small molecule | Adrenergic receptor alpha agonist |
| ergotamine | Agonist | approved | Small molecule | Adrenergic receptor alpha agonist |
| midodrine (proamatine) | Agonist | approved | Small molecule | Adrenergic receptor alpha agonist |
| naphazoline (visine) | Agonist | approved | Small molecule | Adrenergic receptor alpha agonist |
| tetryzoline | Agonist | approved | Small molecule | Adrenergic receptor alpha agonist |
| tramazoline hydrochloride | Agonist | experimental | Small molecule | Adrenergic receptor alpha agonist |
| xylometazoline | Agonist | experimental | Small molecule | Adrenergic receptor alpha agonist |
| aviptadil | Antagonist | experimental | Small molecule | Adrenergic receptor alpha antagonist |
| ergoloid mesylate | Antagonist | approved | Small molecule | Adrenergic receptor alpha antagonist |
| moxisylyte | Antagonist | experimental | Small molecule | Adrenergic receptor alpha antagonist |
| phenoxybenzamine hydrochloride (dibenzyline) | Antagonist | approved | Small molecule | Adrenergic receptor alpha antagonist |
| phentolamine mesylate (regitine) | Antagonist | approved | Small molecule | Adrenergic receptor alpha antagonist |
| rauwolfia alkaloids | Antagonist | approved | Small molecule | Adrenergic receptor alpha antagonist |