← Mechanisms of action
ADRA2A
SINGLE PROTEINHomo sapiens
Preferred name: Alpha-2a adrenergic receptor ChEMBL ↗
Linked proteins
Drugs acting on this target (13)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| regadensoson | Activator | experimental | Small molecule | ADRA2A activator |
| tasipimidine | Agonist | experimental | Small molecule | ADRA2A agonist |
| ciforadenant | Antagonist | experimental | Small molecule | ADRA2A antagonist |
| ct-1500 | Antagonist | experimental | Small molecule | ADRA2A antagonist |
| dzd2269 | Antagonist | experimental | Small molecule | ADRA2A antagonist |
| eos100850 | Antagonist | experimental | Small molecule | ADRA2A antagonist |
| exs21546 | Antagonist | experimental | Small molecule | ADRA2A antagonist |
| inupadenant | Antagonist | experimental | Small molecule | ADRA2A antagonist |
| m1069 | Antagonist | experimental | Small molecule | ADRA2A antagonist |
| mianserin (Tolvon) | Antagonist | experimental | Small molecule | ADRA2A antagonist |
| nir178 | Antagonist | experimental | Small molecule | ADRA2A antagonist |
| idazoxan | Inhibitor | experimental | Small molecule | ADRA2A inhibitor |
| tt-10 | Inhibitor | experimental | Small molecule | ADRA2A inhibitor |