← Mechanisms of action
Adrenergic receptor alpha-1
PROTEIN FAMILYHomo sapiens
Linked proteins
Drugs acting on this target (14)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| alfuzosin (uroxatral) | Agonist | approved | Small molecule | Adrenergic receptor alpha-1 agonist |
| metaraminol (aramine) | Agonist | approved | Small molecule | Adrenergic receptor alpha-1 agonist |
| methoxamine (vasoxyl) | Agonist | approved | Small molecule | Adrenergic receptor alpha-1 agonist |
| phenylephrine (Prefrin) | Agonist | approved | Small molecule | Adrenergic receptor alpha-1 agonist |
| bucindolol | Antagonist | experimental | Small molecule | Adrenergic receptor alpha-1 antagonist |
| Bunazosin (detantol) | Antagonist | experimental | Small molecule | Adrenergic receptor alpha-1 antagonist |
| carvedilol (coreg) | Antagonist | approved | Small molecule | Adrenergic receptor alpha-1 antagonist |
| doxazosin (cardura) | Antagonist | approved | Small molecule | Adrenergic receptor alpha-1 antagonist |
| isoxsuprine | Antagonist | experimental | Small molecule | Adrenergic receptor alpha-1 antagonist |
| prazosin (minipress) | Antagonist | approved | Small molecule | Adrenergic receptor alpha-1 antagonist |
| sertindole (Serdolect) | Antagonist | experimental | Small molecule | Adrenergic receptor alpha-1 antagonist |
| tamsulosin (flomax) | Antagonist | approved | Small molecule | Adrenergic receptor alpha-1 antagonist |
| terazosin (hytrin) | Antagonist | approved | Small molecule | Adrenergic receptor alpha-1 antagonist |
| trimipramine (surmontil) | Antagonist | approved | Small molecule | Adrenergic receptor alpha-1 antagonist |