← Mechanisms of action
ADRA1A
SINGLE PROTEINHomo sapiens
Preferred name: Alpha-1a adrenergic receptor ChEMBL ↗
Linked proteins
Drugs acting on this target (13)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| cst-3056 | Agonist | experimental | Small molecule | ADRA1A agonist |
| da-001 | Agonist | experimental | Small molecule | ADRA1A agonist |
| nrl001 | Agonist | experimental | Small molecule | ADRA1A agonist |
| phenylpropanolamine (Propadrine) | Agonist | withdrawn | Small molecule | ADRA1A agonist |
| xylometazoline | Agonist | experimental | Small molecule | ADRA1A agonist |
| dapiprazole (rev-eyes) | Antagonist | approved | Small molecule | ADRA1A antagonist |
| nicotergoline (Sermion) | Antagonist | experimental | Small molecule | ADRA1A antagonist |
| silodosin (rapaflo) | Antagonist | approved | Small molecule | ADRA1A antagonist |
| talsaclidine | Antagonist | experimental | Small molecule | ADRA1A antagonist |
| tedatioxetine | Antagonist | experimental | Small molecule | ADRA1A antagonist |
| urapidil | Antagonist | experimental | Small molecule | ADRA1A antagonist |
| naftopil (Flivas) | Inhibitor | experimental | Small molecule | ADRA1A inhibitor |
| dabuzalgron | Partial agonist | experimental | Small molecule | ADRA1A partial agonist |