← Mechanisms of action
Tubulin
PROTEIN COMPLEX GROUPHomo sapiens
Linked proteins
- Tubulin beta-4B chain (TUBB4B) ↗
- Tubulin beta-1 chain (TUBB1) ↗
- Tubulin alpha-3C chain (TUBA3C) ↗
- Tubulin alpha-4A chain (TUBA4A) ↗
- Tubulin beta-3 chain (TUBB3) ↗
- Tubulin alpha-1A chain (TUBA1A) ↗
- Tubulin beta-4A chain (TUBB4A) ↗
- Tubulin beta-8 chain (TUBB8) ↗
- Tubulin beta chain (TUBB) ↗
- Tubulin alpha-1B chain (TUBA1B) ↗
- Tubulin alpha-1C chain (TUBA1C) ↗
- Tubulin alpha-3E chain (TUBA3E) ↗
- Tubulin beta-2A chain (TUBB2A) ↗
- Tubulin beta-2B chain (TUBB2B) ↗
- Tubulin beta-6 chain (TUBB6) ↗
Drugs acting on this target (103)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| nL-TUBB4-001 | Antisense inhibitor | experimental | Nucleic acid | Tubulin antisense inhibitor |
| fosbretabulin | Disrupting agent | experimental | Small molecule | Tubulin disrupting agent |
| mpc-6827 | Disrupting agent | experimental | Small molecule | Tubulin disrupting agent |
| rc48-adc | Disrupting agent | experimental | mAb | Tubulin disrupting agent |
| t-900607 | Disrupting agent | experimental | Small molecule | Tubulin disrupting agent |
| abeotaxane | Inhibitor | experimental | Small molecule | Tubulin inhibitor |
| abt-751 | Inhibitor | experimental | Small molecule | Tubulin inhibitor |
| amxi-5001 | Inhibitor | experimental | Small molecule | Tubulin inhibitor |
| anetumab ravtansine | Inhibitor | experimental | mAb | Tubulin inhibitor |
| anhydrovinblastine | Inhibitor | experimental | Small molecule | Tubulin inhibitor |
| asg-5me | Inhibitor | experimental | mAb | Tubulin inhibitor |
| ave-9633 | Inhibitor | experimental | mAb | Tubulin inhibitor |
| bal101553 | Inhibitor | experimental | Small molecule | Tubulin inhibitor |
| batabulin | Inhibitor | experimental | Small molecule | Tubulin inhibitor |
| belantamab mafodotin (TECVAYLI) | Inhibitor | approved | mAb | Tubulin inhibitor |
| benzimidazole | Inhibitor | experimental | Small molecule | Tubulin inhibitor |
| biib-015 | Inhibitor | experimental | mAb | Tubulin inhibitor |
| bivatuzumab mertansine | Inhibitor | experimental | mAb | Tubulin inhibitor |
| bms-184476 | Inhibitor | experimental | Small molecule | Tubulin inhibitor |
| bms-188797 | Inhibitor | experimental | Small molecule | Tubulin inhibitor |
| bms-275183 | Inhibitor | experimental | Small molecule | Tubulin inhibitor |
| bnc 105p | Inhibitor | experimental | Small molecule | Tubulin inhibitor |
| brentuximab vedotin (adcetris) | Inhibitor | approved | mAb | Tubulin inhibitor |
| cabazitaxel (jevtana kit) | Inhibitor | approved | Small molecule | Tubulin inhibitor |
| cantuzumab mertansine | Inhibitor | experimental | mAb | Tubulin inhibitor |
| cantuzumab ravtansine | Inhibitor | experimental | mAb | Tubulin inhibitor |
| cci-001 | Inhibitor | experimental | Small molecule | Tubulin inhibitor |
| ckd-516 | Inhibitor | experimental | Small molecule | Tubulin inhibitor |
| colchicine (colbenemid) | Inhibitor | approved | Small molecule | Tubulin inhibitor |
| coltuximab ravtansine | Inhibitor | experimental | mAb | Tubulin inhibitor |
| crinobulin | Inhibitor | experimental | Small molecule | Tubulin inhibitor |
| cyt997 | Inhibitor | experimental | Small molecule | Tubulin inhibitor |
| depatuxizumab mafodotin | Inhibitor | experimental | mAb | Tubulin inhibitor |
| docetaxel (taxotere) | Inhibitor | approved | Small molecule | Tubulin inhibitor |
| e7130 | Inhibitor | experimental | Small molecule | Tubulin inhibitor |
| e7974 | Inhibitor | experimental | Small molecule | Tubulin inhibitor |
| ec1169 | Inhibitor | experimental | Small molecule | Tubulin inhibitor |
| ec1456 | Inhibitor | experimental | Small molecule | Tubulin inhibitor |
| enfortumab vedotin (Padcev) | Inhibitor | approved | mAb | Tubulin inhibitor |
| epc2407 | Inhibitor | experimental | Small molecule | Tubulin inhibitor |
| epothilone | Inhibitor | experimental | Small molecule | Tubulin inhibitor |
| eribulin (halaven) | Inhibitor | approved | Small molecule | Tubulin inhibitor |
| fluorapacin | Inhibitor | experimental | Small molecule | Tubulin inhibitor |
| fosbretabulin | Inhibitor | experimental | Small molecule | Tubulin inhibitor |
| glembatumumab vedotin | Inhibitor | experimental | mAb | Tubulin inhibitor |
| imgn-388 | Inhibitor | experimental | mAb | Tubulin inhibitor |
| indatuximab ravtansine | Inhibitor | experimental | mAb | Tubulin inhibitor |
| indibulin | Inhibitor | experimental | Small molecule | Tubulin inhibitor |
| ixabepilone (ixempra) | Inhibitor | approved | Small molecule | Tubulin inhibitor |
| kosn-1724 | Inhibitor | experimental | Small molecule | Tubulin inhibitor |
| ladiratuzumab vedotin | Inhibitor | experimental | mAb | Tubulin inhibitor |
| lorvotuzumab mertansine | Inhibitor | experimental | mAb | Tubulin inhibitor |
| Losatuxizumab vedotin | Inhibitor | experimental | mAb | Tubulin inhibitor |
| milataxel | Inhibitor | experimental | Small molecule | Tubulin inhibitor |
| mirvetuximab soravtansine (Elahere) | Inhibitor | approved | mAb | Tubulin inhibitor |
| mln-2704 | Inhibitor | experimental | mAb | Tubulin inhibitor |
| mpc6827 | Inhibitor | experimental | Small molecule | Tubulin inhibitor |
| noscapine | Inhibitor | experimental | Small molecule | Tubulin inhibitor |
| nov120401 | Inhibitor | experimental | Small molecule | Tubulin inhibitor |
| oc-10x | Inhibitor | experimental | Small molecule | Tubulin inhibitor |
| ombrabulin | Inhibitor | experimental | Small molecule | Tubulin inhibitor |
| paclitaxel (taxol) | Inhibitor | approved | Small molecule | Tubulin inhibitor |
| pf-06263507 | Inhibitor | experimental | mAb | Tubulin inhibitor |
| plinabulin | Inhibitor | experimental | Small molecule | Tubulin inhibitor |
| pm060184 | Inhibitor | experimental | Small molecule | Tubulin inhibitor |
| pm534 | Inhibitor | experimental | Small molecule | Tubulin inhibitor |
| podophyllin | Inhibitor | experimental | Biological | Tubulin inhibitor |
| polatuzumab vedotin (Polivy) | Inhibitor | approved | mAb | Tubulin inhibitor |
| ptc596 | Inhibitor | experimental | Small molecule | Tubulin inhibitor |
| rg-7598 | Inhibitor | experimental | mAb | Tubulin inhibitor |
| rg-7600 | Inhibitor | experimental | mAb | Tubulin inhibitor |
| rg-7636 | Inhibitor | experimental | mAb | Tubulin inhibitor |
| sabizabulin | Inhibitor | experimental | Small molecule | Tubulin inhibitor |
| sar408701 | Inhibitor | experimental | mAb | Tubulin inhibitor |
| sar566658 | Inhibitor | experimental | mAb | Tubulin inhibitor |
| scb01a | Inhibitor | experimental | Small molecule | Tubulin inhibitor |
| simotaxel | Inhibitor | experimental | Small molecule | Tubulin inhibitor |
| soblidotin | Inhibitor | experimental | Small molecule | Tubulin inhibitor |
| sofituzumab vedotin | Inhibitor | experimental | mAb | Tubulin inhibitor |
| ssr97225 | Inhibitor | experimental | Small molecule | Tubulin inhibitor |
| sta-5312 | Inhibitor | experimental | Small molecule | Tubulin inhibitor |
| t-900607 | Inhibitor | experimental | Small molecule | Tubulin inhibitor |
| tasidotin | Inhibitor | experimental | Small molecule | Tubulin inhibitor |
| telisotuzumab vedodin (Emrelis) | Inhibitor | approved | mAb | Tubulin inhibitor |
| tesetaxel | Inhibitor | experimental | Small molecule | Tubulin inhibitor |
| tisotumab vedotin (TIVDAK) | Inhibitor | approved | mAb | Tubulin inhibitor |
| trastuzumab emtansine (kadcyla) | Inhibitor | approved | mAb | Tubulin inhibitor |
| verobulin (Azixa) | Inhibitor | experimental | Small molecule | Tubulin inhibitor |
| vinblastine (velban) | Inhibitor | approved | Small molecule | Tubulin inhibitor |
| vincristine (oncovin) | Inhibitor | approved | Small molecule | Tubulin inhibitor |
| vindesine (Eldisine) | Inhibitor | experimental | Small molecule | Tubulin inhibitor |
| vinflunine | Inhibitor | experimental | Small molecule | Tubulin inhibitor |
| vinorelbine (navelbine) | Inhibitor | approved | Small molecule | Tubulin inhibitor |
| wh002 | Inhibitor | experimental | Small molecule | Tubulin inhibitor |
| zd6126 | Inhibitor | experimental | Small molecule | Tubulin inhibitor |
| bms-275183 | Stabiliser | experimental | Small molecule | Tubulin stabiliser |
| davunetide | Stabiliser | experimental | Peptide | Tubulin stabiliser |
| docetaxel (taxotere) | Stabiliser | approved | Small molecule | Tubulin stabiliser |
| epothilone | Stabiliser | experimental | Small molecule | Tubulin stabiliser |
| kos-1584 | Stabiliser | experimental | Botanical | Tubulin stabiliser |
| larotaxel | Stabiliser | experimental | Small molecule | Tubulin stabiliser |
| paclitaxel (taxol) | Stabiliser | approved | Small molecule | Tubulin stabiliser |
| sagopilone | Stabiliser | experimental | Small molecule | Tubulin stabiliser |