← Mechanisms of action
Bacterial DNA gyrase
PROTEIN COMPLEXBacteria
Linked proteins
Drugs acting on this target (24)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| nalidixic acid (neggram) | Antagonist | approved | Small molecule | Bacterial DNA gyrase antagonist |
| norfloxacin (noroxin) | Antagonist | approved | Small molecule | Bacterial DNA gyrase antagonist |
| sparfloxacin (zagam) | Antagonist | approved | Small molecule | Bacterial DNA gyrase antagonist |
| trovafloxacin (trovan) | Antagonist | approved | Small molecule | Bacterial DNA gyrase antagonist |
| Acorafloxacin | Inhibitor | experimental | Small molecule | Bacterial DNA gyrase inhibitor |
| alatrofloxacin (trovan) | Inhibitor | approved | Small molecule | Bacterial DNA gyrase inhibitor |
| besifloxacin (besivance) | Inhibitor | approved | Small molecule | Bacterial DNA gyrase inhibitor |
| cinoxacin (cinobac) | Inhibitor | approved | Small molecule | Bacterial DNA gyrase inhibitor |
| ciprofloxacin (cipro) | Inhibitor | approved | Small molecule | Bacterial DNA gyrase inhibitor |
| delafloxacin meglumine (baxdela) | Inhibitor | approved | Small molecule | Bacterial DNA gyrase inhibitor |
| gepotidacin | Inhibitor | approved | Small molecule | Bacterial DNA gyrase inhibitor |
| levonadifloxacin | Inhibitor | experimental | Small molecule | Bacterial DNA gyrase inhibitor |
| lomefloxacin (maxaquin) | Inhibitor | approved | Small molecule | Bacterial DNA gyrase inhibitor |
| moxifloxacin (avelox) | Inhibitor | approved | Small molecule | Bacterial DNA gyrase inhibitor |
| nemonoxacin | Inhibitor | experimental | Small molecule | Bacterial DNA gyrase inhibitor |
| novobiocin (albamycin) | Inhibitor | approved | Small molecule | Bacterial DNA gyrase inhibitor |
| ofloxacin (floxin) | Inhibitor | approved | Small molecule | Bacterial DNA gyrase inhibitor |
| pazufloxacin | Inhibitor | experimental | Small molecule | Bacterial DNA gyrase inhibitor |
| pefloxacine | Inhibitor | experimental | Small molecule | Bacterial DNA gyrase inhibitor |
| prulifloxacin | Inhibitor | experimental | Small molecule | Bacterial DNA gyrase inhibitor |
| sitafloxacin | Inhibitor | experimental | Small molecule | Bacterial DNA gyrase inhibitor |
| temafloxacin (Omniflox) | Inhibitor | approved | Small molecule | Bacterial DNA gyrase inhibitor |
| trovafloxacin (trovan) | Inhibitor | approved | Small molecule | Bacterial DNA gyrase inhibitor |
| zabofloxacin | Inhibitor | experimental | Small molecule | Bacterial DNA gyrase inhibitor |