← Mechanisms of action

DNA topoisomerase II

PROTEIN FAMILYHomo sapiens

Linked proteins

Drugs acting on this target (21)

Active Pharmaceutical Ingredient Mechanism Type Approval Status API Type Mechanism of Action
aminocamptothecinInhibitorexperimentalSmall moleculeDNA topoisomerase II inhibitor
amonafideInhibitorexperimentalSmall moleculeDNA topoisomerase II inhibitor
amsacrineInhibitorexperimentalSmall moleculeDNA topoisomerase II inhibitor
ava6000InhibitorexperimentalSmall moleculeDNA topoisomerase II inhibitor
banoxantroneInhibitorexperimentalSmall moleculeDNA topoisomerase II inhibitor
becatecarinInhibitorexperimentalSmall moleculeDNA topoisomerase II inhibitor
CamsirubicinInhibitorexperimentalSmall moleculeDNA topoisomerase II inhibitor
daniquidoneInhibitorexperimentalSmall moleculeDNA topoisomerase II inhibitor
dexrazoxane (zinecard)InhibitorapprovedSmall moleculeDNA topoisomerase II inhibitor
etoposide (vepesid)InhibitorapprovedSmall moleculeDNA topoisomerase II inhibitor
intoplicineInhibitorexperimentalSmall moleculeDNA topoisomerase II inhibitor
mk-2248InhibitorexperimentalSmall moleculeDNA topoisomerase II inhibitor
nsc-645809InhibitorexperimentalSmall moleculeDNA topoisomerase II inhibitor
pazufloxacinInhibitorexperimentalSmall moleculeDNA topoisomerase II inhibitor
pirarubicinInhibitorexperimentalSmall moleculeDNA topoisomerase II inhibitor
rta 744InhibitorexperimentalSmall moleculeDNA topoisomerase II inhibitor
sabarubicinInhibitorexperimentalSmall moleculeDNA topoisomerase II inhibitor
sq3370InhibitorexperimentalSmall moleculeDNA topoisomerase II inhibitor
teniposide (vumon)InhibitorapprovedSmall moleculeDNA topoisomerase II inhibitor
vosaroxinInhibitorexperimentalSmall moleculeDNA topoisomerase II inhibitor
xk469InhibitorexperimentalSmall moleculeDNA topoisomerase II inhibitor