CDEK
← Mechanisms of action

AR

SINGLE PROTEINHomo sapiens
Preferred name: Androgen Receptor ChEMBL ↗

Linked proteins

Drugs acting on this target (93)

Active Pharmaceutical Ingredient Mechanism Type ▲ Approval Status API Type Mechanism of Action
17-a-methyl-etioallocholan-17b-ol-3-hydroxyimineAgonistexperimentalSmall moleculeAR agonist
cr1447AgonistexperimentalSmall moleculeAR agonist
danazol (danocrine)AgonistapprovedSmall moleculeAR agonist
drostanolone (drolban)AgonistapprovedSmall moleculeAR agonist
ethylestrenol (maxibolin)AgonistapprovedSmall moleculeAR agonist
fluoxymesteroneAgonistapprovedSmall moleculeAR agonist
gw-501516 (Cardarine)AgonistexperimentalSmall moleculeAR agonist
methyltestosterone (testred)AgonistapprovedSmall moleculeAR agonist
nandrolone phenpropionate (Durabolin)AgonistapprovedSmall moleculeAR agonist
Norethandrolone (Pronabol)AgonistexperimentalSmall moleculeAR agonist
oxandrolone (oxandrin)AgonistapprovedSmall moleculeAR agonist
oxymetholone (anadrol-50)AgonistapprovedSmall moleculeAR agonist
progestinAgonistexperimentalSmall moleculeAR agonist
stanoloneAgonistexperimentalSmall moleculeAR agonist
stanozolol (winstrol)AgonistapprovedSmall moleculeAR agonist
testosterone (delatestryl)AgonistapprovedSmall moleculeAR agonist
trestoloneAgonistexperimentalSmall moleculeAR agonist
abiraterone (zytiga)AntagonistapprovedSmall moleculeAR antagonist
apalutamide (erleada)AntagonistapprovedSmall moleculeAR antagonist
apc-100AntagonistexperimentalSmall moleculeAR antagonist
bay1161116AntagonistexperimentalSmall moleculeAR antagonist
bicalutamide (casodex)AntagonistapprovedSmall moleculeAR antagonist
clascoterone (Winlevi)AntagonistapprovedSmall moleculeAR antagonist
cyprovironAntagonistexperimentalSmall moleculeAR antagonist
darolutamide (Nubeqa)AntagonistapprovedSmall moleculeAR antagonist
enzalutamide (xtandi)AntagonistapprovedSmall moleculeAR antagonist
flutamide (eulexin)AntagonistapprovedSmall moleculeAR antagonist
ft-7051AntagonistexperimentalSmall moleculeAR antagonist
galeteroneAntagonistexperimentalSmall moleculeAR antagonist
kx- 826AntagonistexperimentalSmall moleculeandrogen receptor
kx0826AntagonistexperimentalSmall moleculeAR antagonist
nilutamide (nilandron)AntagonistapprovedSmall moleculeAR antagonist
p2613422AntagonistexperimentalSmall moleculeAR antagonist
proxalutamideAntagonistexperimentalPeptideAR antagonist
RezvilutamideAntagonistexperimentalSmall moleculeAndrogen Receptor antagonist
seviteronelAntagonistexperimentalSmall moleculeAndrogen Receptor antagonist
tqb3720AntagonistexperimentalSmall moleculeAR antagonist
trc253AntagonistexperimentalSmall moleculeAR antagonist
sxl01Antisense inhibitorexperimentalNucleic acidAR antisense inhibitor
18 F-Fluoro-5α-DihydrotestosteroneBinding agentexperimentalSmall moleculeAR binding agent
ac176DegraderexperimentalSmall moleculeAndrogen Receptor degrader
ah-001DegraderexperimentalSmall moleculeAR degrader
arv-110DegraderexperimentalSmall moleculeAR degrader
arv-766DegraderexperimentalSmall moleculeAR degrader
azd9750DegraderexperimentalSmall moleculeAR degrader
bn104DegraderexperimentalSmall moleculeAR degrader
cc-94676DegraderexperimentalSmall moleculeAR degrader
DimethylcurcuminDegraderexperimentalSmall moleculeAndrogen Receptor degrader
gt-220fDegraderexperimentalSmall moleculeAR degrader
gt20029DegraderexperimentalSmall moleculeandrogen receptor
hp518DegraderexperimentalSmall moleculeandrogen receptor
hrs-5041DegraderexperimentalSmall moleculeAR degrader
luxdegalutamideDegraderexperimentalSmall moleculeAR degrader
tqb3201DegraderexperimentalSmall moleculeAR degrader
ptvg-arImmunity, activeexperimentalVaccineAR immunity, active
11betamethyl nortestosterone dodecylcarbonateInhibitorexperimentalSmall moleculeAR inhibitor
ar51InhibitorexperimentalVaccineAR inhibitor
bay2688901InhibitorexperimentalSmall moleculeAR inhibitor
bms-986409InhibitorexperimentalSmall moleculeAR inhibitor
bms-986410InhibitorexperimentalSmall moleculeAR inhibitor
bms641988InhibitorexperimentalSmall moleculeAR inhibitor
Cyproterone (Androcur)InhibitorexperimentalSmall moleculeAR inhibitor
deuterated enzalutamideInhibitorexperimentalSmall moleculeAR inhibitor
epi-506InhibitorexperimentalSmall moleculeAR inhibitor
epi-7386InhibitorexperimentalSmall moleculeAR inhibitor
hld-0915InhibitorexperimentalSmall moleculeAR inhibitor
HydroxyflutamideInhibitorexperimentalSmall moleculeAR inhibitor
odm-204InhibitorexperimentalSmall moleculeAR inhibitor
onc1-0013bInhibitorexperimentalSmall moleculeAR inhibitor
onct-534InhibitorexperimentalSmall moleculeAR inhibitor
pf-06260414InhibitorexperimentalSmall moleculeAR inhibitor
qlg1080InhibitorexperimentalSmall moleculeAR inhibitor
RezvilutamideInhibitorexperimentalSmall moleculeAR inhibitor
sb-509InhibitorexperimentalSmall moleculeAR inhibitor
shr 3680InhibitorexperimentalSmall moleculeAR inhibitor
tas3681InhibitorexperimentalSmall moleculeAR inhibitor
azd-3514ModulatorexperimentalSmall moleculeAR modulator
enobosarmModulatorexperimentalSmall moleculeAR modulator
glpg-0492ModulatorexperimentalSmall moleculeAR modulator
gsk2849466ModulatorexperimentalSmall moleculeAR modulator
gsk2881078ModulatorexperimentalSmall moleculeAR modulator
gsk971086ModulatorexperimentalSmall moleculeAR modulator
he3235ModulatorexperimentalSmall moleculeAR modulator
lgd-4033ModulatorexperimentalSmall moleculeAR modulator
lgd2941ModulatorexperimentalSmall moleculeAR modulator
ly-2452473ModulatorexperimentalSmall moleculeAR modulator
mk0773ModulatorexperimentalSmall moleculeAR modulator
nido-361ModulatorexperimentalSmall moleculeAR modulator
opk-88004ModulatorexperimentalSmall moleculeAR modulator
rad140ModulatorexperimentalSmall moleculeAR modulator
tetrahydrogestrinoneModulatorexperimentalSmall moleculeAR modulator
VosilasarmModulatorexperimentalSmall moleculeAR modulator
fluorofuranylnorprogesteroneRadiopharmaceuticalexperimentalSmall moleculeAR radiopharmaceutical