← Mechanisms of action
HTR1A
SINGLE PROTEINHomo sapiens
Preferred name: Serotonin 1a (5-HT1a) receptor ChEMBL ↗
Linked proteins
Drugs acting on this target (42)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| befiradol | Agonist | experimental | Small molecule | HTR1A agonist |
| DSP-9632P | Agonist | experimental | Small molecule | HTR1A agonist |
| eltoprazine | Agonist | experimental | Small molecule | HTR1A agonist |
| enx-205 | Agonist | experimental | Small molecule | HTR1A agonist |
| ergoloid mesylate | Agonist | approved | Small molecule | HTR1A agonist |
| f13640 | Agonist | experimental | Small molecule | HTR1A agonist |
| gepirone monohydrochloride (Exxua) | Agonist | approved | Small molecule | Serotonin 1a (5-HT1a) receptor agonist |
| lisuride (Dopergin) | Agonist | experimental | Small molecule | HTR1A agonist |
| lysergic acid diethylamide | Agonist | experimental | Small molecule | HTR1A agonist |
| Methylergonovine | Agonist | experimental | Biological | HTR1A agonist |
| mn-305 | Agonist | experimental | Small molecule | HTR1A agonist |
| naluzotan | Agonist | experimental | Small molecule | HTR1A agonist |
| pardoprunox | Agonist | experimental | Small molecule | HTR1A agonist |
| piclozotan | Agonist | experimental | Small molecule | HTR1A agonist |
| repinotan | Agonist | experimental | Small molecule | HTR1A agonist |
| sarizotan | Agonist | experimental | Small molecule | HTR1A agonist |
| slv-313 | Agonist | experimental | Small molecule | HTR1A agonist |
| Ulotaront | Agonist | experimental | Small molecule | HTR1A agonist |
| urapidil | Agonist | experimental | Small molecule | HTR1A agonist |
| uropidil | Agonist | experimental | Small molecule | HTR1A agonist |
| vortioxetine (trintellix) | Agonist | approved | Small molecule | HTR1A agonist |
| xaliproden hydrochloride | Agonist | experimental | Small molecule | HTR1A agonist |
| ati-9242 | Antagonist | experimental | Small molecule | HTR1A antagonist |
| dosulepin (Prothiaden) | Antagonist | experimental | Small molecule | HTR1A antagonist |
| du125530 | Antagonist | experimental | Small molecule | HTR1A antagonist |
| gsk163090 | Antagonist | experimental | Small molecule | HTR1A antagonist |
| gsk958108 | Antagonist | experimental | Small molecule | HTR1A antagonist |
| lecozotan | Antagonist | experimental | Small molecule | HTR1A antagonist |
| mppf | Antagonist | experimental | Small molecule | HTR1A antagonist |
| phenpropamine | Antagonist | experimental | Small molecule | HTR1A antagonist |
| robalzotan | Antagonist | experimental | Small molecule | HTR1A antagonist |
| min-117 | Inhibitor | experimental | Small molecule | HTR1A inhibitor |
| aripiprazole (abilify) | Partial agonist | approved | Small molecule | HTR1A partial agonist |
| bifeprunoxum | Partial agonist | experimental | Small molecule | HTR1A partial agonist |
| brexpiprazole (rexulti) | Partial agonist | approved | Small molecule | HTR1A partial agonist |
| Brilaroxazine | Partial agonist | experimental | Small molecule | HTR1A partial agonist |
| buspirone (buspar) | Partial agonist | approved | Small molecule | HTR1A partial agonist |
| dsp-1053 | Partial agonist | experimental | Small molecule | HTR1A partial agonist |
| gepirone monohydrochloride (Exxua) | Partial agonist | approved | Small molecule | HTR1A partial agonist |
| methysergide (sansert) | Partial agonist | approved | Small molecule | HTR1A partial agonist |
| tandospirone | Partial agonist | experimental | Small molecule | HTR1A partial agonist |
| vilazodone (viibryd) | Partial agonist | approved | Small molecule | HTR1A partial agonist |