← Mechanisms of action
TACR1
SINGLE PROTEINHomo sapiens
Preferred name: Neurokinin 1 receptor ChEMBL ↗
Linked proteins
Drugs acting on this target (26)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| aprepitant (Emend) | Antagonist | approved | Small molecule | TACR1 antagonist |
| av608 | Antagonist | experimental | Small molecule | TACR1 antagonist |
| Casopitant (zunrisa) | Antagonist | experimental | Small molecule | TACR1 antagonist |
| dnk333 | Antagonist | experimental | Small molecule | TACR1 antagonist |
| elinzanetant | Antagonist | approved | Small molecule | TACR1 antagonist |
| ezlopitant | Antagonist | experimental | Small molecule | TACR1 antagonist |
| figopitant | Antagonist | experimental | Small molecule | TACR1 antagonist |
| fosnetupitant (Akynzeo) | Antagonist | approved | Small molecule | Neurokinin 1 receptor antagonist |
| gr2301 | Antagonist | experimental | Small molecule | TACR1 antagonist |
| gsk1144814 | Antagonist | experimental | Small molecule | TACR1 antagonist |
| gsk424887 | Antagonist | experimental | Small molecule | TACR1 antagonist |
| netupitant (Akynzeo) | Antagonist | approved | Small molecule | TACR1 antagonist |
| nt-814 | Antagonist | experimental | Small molecule | TACR1 antagonist |
| orvepitant | Antagonist | experimental | Small molecule | TACR1 antagonist |
| rolapitant (varubi) | Antagonist | approved | Small molecule | TACR1 antagonist |
| serlopitant | Antagonist | experimental | Small molecule | TACR1 antagonist |
| ssr240600 | Antagonist | experimental | Small molecule | TACR1 antagonist |
| tradipitant | Antagonist | approved | Small molecule | TACR1 antagonist |
| vestipitant mesylate | Antagonist | experimental | Small molecule | TACR1 antagonist |
| vofopitant | Antagonist | experimental | Small molecule | TACR1 antagonist |
| gsk206136 | Inhibitor | experimental | Small molecule | TACR1 inhibitor |
| m516102 | Inhibitor | experimental | Small molecule | TACR1 inhibitor |
| slv317 | Inhibitor | experimental | Small molecule | TACR1 inhibitor |
| substance p | Inhibitor | experimental | Small molecule | TACR1 inhibitor |
| thonzonium bromide | Inhibitor | approved | Small molecule | TACR1 inhibitor |
| vestipitant | Inhibitor | experimental | Small molecule | TACR1 inhibitor |