peficitinib

Trade name: Vonjo

Small moleculeexperimental

Peficitinib is a pharmaceutical drug used for the treatment of rheumatoid arthritis. It belongs to the class of drugs known as Janus kinase inhibitors. — Wikipedia

Chemistry & pharmacology

Loading structure…

SMILES

NC(=O)c1cnc2[nH]ccc2c1N[C@@H]1[C@@H]2CC3C[C@H]1C[C@@](O)(C3)C2
Mol. weight
326.4 g/mol
Lipinski Ro5
Pass
Rule of 3
No
Chirality
Racemic Mixture
Inorganic
No
Polymer
No
Delivery
Oral

Oral

Yes

Parenteral

No

Topical

No

Sources

Also known as

  • 4-((5-hydroxy-2-adamantyl)amino)-1h-pyrrolo(2,3-b)pyridine-5-carboxamide
  • asp015k
  • asp015k
  • asp015k
  • asp015k
  • asp-015k
  • asp-015k
  • jnj-54781532
  • jnj-54781532
  • peficitinib
  • peficitinib
  • peficitinib

Clinical trials

NCT IDPhaseStart dateSponsor(s)
NCT04143477Phase 1Oct 31, 2019Astellas
NCT03660059Phase 3Sep 30, 2018Astellas
NCT02760342Phase 1May 1, 2016Astellas
NCT02603497Phase 1Nov 1, 2015Astellas
NCT02586194Phase 1Nov 1, 2015Astellas
NCT02531191Phase 1Jun 1, 2015Astellas
NCT02305849Phase 3Jul 25, 2014Astellas
NCT02308163Phase 3Jul 1, 2014Astellas
NCT02117505Phase 1Apr 1, 2014Johnson and Johnson
NCT02141425Phase 1Mar 1, 2014Astellas, Janssen Pharmaceutica NV
NCT01959282Phase 2Nov 1, 2013Johnson and Johnson
NCT02111317Phase 1Oct 1, 2013Astellas, Janssen Pharmaceutica NV
NCT01959399Phase 1May 1, 2013Astellas, Janssen Pharmaceutica NV
NCT01929577Phase 1May 1, 2013Astellas, Janssen Pharmaceutica NV
NCT01711814Phase 2Sep 1, 2012Astellas, Janssen Pharmaceutica NV
NCT01638013Phase 3Jun 13, 2012Astellas
NCT01686217Phase 1Jun 1, 2012Astellas
NCT01554696Phase 2Jun 1, 2012Astellas
NCT01565655Phase 2Jun 1, 2012Astellas
NCT01649999Phase 2Feb 1, 2012Astellas
Showing 20 of 34 trials
Page 1 / 2

Organizations

Research & Development (4)

OrganizationOrg typeTrialsAs lead sponsorPhasesEarliest year
AstellasFor profit313132008
Janssen Pharmaceutica NVFor profit5022012
Johnson and JohnsonFor profit2222013
PfizerFor profit1112011
4 organizations
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