← Mechanisms of action

JAK3

SINGLE PROTEINHomo sapiens
Preferred name: Tyrosine-protein kinase JAK3 ChEMBL ↗

Linked proteins

Drugs acting on this target (27)

Active Pharmaceutical Ingredient Mechanism Type Approval Status API Type Mechanism of Action
at9283InhibitorexperimentalSmall moleculeJAK3 inhibitor
ati-2138InhibitorexperimentalSmall moleculeJAK3 inhibitor
ati-50002InhibitorexperimentalSmall moleculeJAK3 inhibitor
ati-501InhibitorexperimentalSmall moleculeJAK3 inhibitor
cerdulatinibInhibitorexperimentalSmall moleculeJAK3 inhibitor
cs12192InhibitorexperimentalSmall moleculeJAK3 inhibitor
decernotinibInhibitorexperimentalSmall moleculeJAK3 inhibitor
delgocitinib (Anzupgo)InhibitorapprovedSmall moleculeJAK3 inhibitor
deuruxolitinibInhibitorapprovedSmall moleculeTyrosine-protein kinase JAK3 inhibitor
dwp212525InhibitorexperimentalSmall moleculeJAK3 inhibitor
filgotinib (Jyseleca)InhibitorexperimentalSmall moleculeTyrosine-protein kinase JAK3 inhibitor
IfidancitinibInhibitorexperimentalSmall moleculeJAK3 inhibitor
max-40070InhibitorexperimentalSmall moleculeJAK3 inhibitor
or-101InhibitorexperimentalSmall moleculeJAK3 inhibitor
ost-122InhibitorexperimentalSmall moleculeJAK3 inhibitor
pf06263276InhibitorexperimentalSmall moleculeJAK3 inhibitor
r-333InhibitorexperimentalSmall moleculeJAK3 inhibitor
r-348InhibitorexperimentalSmall moleculeJAK3 inhibitor
r348InhibitorexperimentalSmall moleculeJAK3 inhibitor
r932333InhibitorexperimentalSmall moleculeJAK3 inhibitor
ritlecitinib (Litfulo)InhibitorapprovedSmall moleculeJAK3 inhibitor
td-5202InhibitorexperimentalSmall moleculeJAK3 inhibitor
td-8236InhibitorexperimentalSmall moleculeJAK3 inhibitor
tofacitinib (xeljanz)InhibitorapprovedSmall moleculeJAK3 inhibitor
tricetamideInhibitorexperimentalSmall moleculeJAK3 inhibitor
whi-p131InhibitorexperimentalSmall moleculeJAK3 inhibitor
zl-82InhibitorexperimentalSmall moleculeJAK3 inhibitor