← Mechanisms of action

TYK2

SINGLE PROTEINHomo sapiens
Preferred name: Tyrosine-protein kinase TYK2 ChEMBL ↗

Linked proteins

Drugs acting on this target (41)

Active Pharmaceutical Ingredient Mechanism Type Approval Status API Type Mechanism of Action
esk-001AntagonistexperimentalSmall moleculeTyk2
icp-332AntagonistexperimentalSmall moleculeTYK2
icp-488AntagonistexperimentalSmall moleculeTYK2
a-005InhibitorexperimentalSmall moleculeTYK2 inhibitor
a51r2InhibitorexperimentalSmall moleculeTYK2 inhibitor
abbv-722InhibitorexperimentalSmall moleculeTYK2 inhibitor
bgb-23339InhibitorexperimentalSmall moleculeTYK2 inhibitor
bhv-8000InhibitorexperimentalSmall moleculeTYK2 inhibitor
blkr201InhibitorexperimentalSmall moleculeTYK2 inhibitor
bms-986202InhibitorexperimentalSmall moleculeTYK2 inhibitor
bms-986482InhibitorexperimentalSmall moleculeTYK2 inhibitor
bms-986482InhibitorexperimentalSmall moleculeTYK2 inhibitor
BrepocitinibInhibitorexperimentalSmall moleculeTYK2 inhibitor
cerdulatinibInhibitorexperimentalSmall moleculeTYK2 inhibitor
cms-d001InhibitorexperimentalSmall moleculeTYK2 inhibitor
cs32582InhibitorexperimentalSmall moleculeTYK2 inhibitor
d-2570InhibitorexperimentalSmall moleculeTYK2 inhibitor
deuruxolitinibInhibitorapprovedSmall moleculeTyrosine-protein kinase TYK2 inhibitor
filgotinib (Jyseleca)InhibitorexperimentalSmall moleculeTyrosine-protein kinase TYK2 inhibitor
glpg3121InhibitorexperimentalSmall moleculeTYK2 inhibitor
glpg3667InhibitorexperimentalSmall moleculeTYK2 inhibitor
hs-10374InhibitorexperimentalSmall moleculeTYK2 inhibitor
max-40070InhibitorexperimentalSmall moleculeTYK2 inhibitor
neu-627InhibitorexperimentalSmall moleculeTYK2 inhibitor
ost-122InhibitorexperimentalSmall moleculeTYK2 inhibitor
pf-06826647InhibitorexperimentalSmall moleculeTYK2 inhibitor
pf06263276InhibitorexperimentalSmall moleculeTYK2 inhibitor
qy201InhibitorexperimentalSmall moleculeTYK2 inhibitor
syhx 1901InhibitorexperimentalSmall moleculeTYK2 inhibitor
syhx1901InhibitorexperimentalSmall moleculeTYK2 inhibitor
tdm-180935InhibitorexperimentalSmall moleculeTYK2 inhibitor
tll-018InhibitorexperimentalSmall moleculeTYK2 inhibitor
tll018InhibitorexperimentalSmall moleculeTYK2 inhibitor
tqh3906InhibitorexperimentalSmall moleculeTYK2 inhibitor
ty-2136bInhibitorexperimentalSmall moleculeTYK2 inhibitor
vtx958InhibitorexperimentalSmall moleculeTYK2 inhibitor
vvn461InhibitorexperimentalSmall moleculeTYK2 inhibitor
wd-890InhibitorexperimentalSmall moleculeTYK2 inhibitor
wd-910InhibitorexperimentalSmall moleculeTYK2 inhibitor
zasocitinibInhibitorexperimentalSmall moleculeTYK2 inhibitor
deucravacitinib (Sotkyktu)Negative allosteric modulatorapprovedSmall moleculeTyrosine-protein kinase TYK2 negative allosteric modulator