← Mechanisms of action
GABA-A receptor
PROTEIN COMPLEX GROUPSarcoptes scabiei
Linked proteins
Drugs acting on this target (11)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| remimazolam (Byfavo) | Activator | approved | Small molecule | GABA-A receptor activator |
| elb-139 | Agonist | experimental | Small molecule | GABA-A receptor agonist |
| fospropofol (lusedra) | Agonist | approved | Small molecule | GABA-A receptor agonist |
| secobarbital (seconal) | Agonist | approved | Small molecule | GABA-A receptor agonist |
| stiripentol (diacomit) | Agonist | approved | Small molecule | GABA-A receptor agonist |
| brexanolone (Zulresso) | Allosteric antagonist | approved | Small molecule | GABA-A receptor allosteric antagonist |
| lorazepam (ativan) | Allosteric antagonist | approved | Small molecule | GABA-A receptor allosteric antagonist |
| phenobarbital (Luminal) | Allosteric antagonist | approved | Small molecule | GABA-A receptor allosteric antagonist |
| meprobamate (equanil) | Binding agent | approved | Small molecule | GABA-A receptor binding agent |
| lotilaner (xdemvy) | Inhibitor | approved | Small molecule | GABA-A receptor inhibitor |
| lindane (kwell) | Negative allosteric modulator | approved | Small molecule | GABA-A receptor negative allosteric modulator |