← Mechanisms of action
ADRB1
SINGLE PROTEINHomo sapiens
Preferred name: Beta-1 adrenergic receptor ChEMBL ↗
Linked proteins
Drugs acting on this target (33)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| Etafedrine | Activator | experimental | Small molecule | ADRB1 activator |
| dobutamine (dobutrex) | Agonist | approved | Small molecule | ADRB1 agonist |
| dopamine (intropin) | Agonist | approved | Small molecule | ADRB1 agonist |
| foslevodopa (VYALEV) | Agonist | approved | Small molecule | Beta-1 adrenergic receptor agonist |
| acebutolol (sectral) | Antagonist | approved | Small molecule | ADRB1 antagonist |
| atenolol (tenormin) | Antagonist | approved | Small molecule | ADRB1 antagonist |
| betaxolol (kerlone) | Antagonist | approved | Small molecule | ADRB1 antagonist |
| bisoprolol (zebeta) | Antagonist | approved | Small molecule | ADRB1 antagonist |
| bucindolol | Antagonist | experimental | Small molecule | ADRB1 antagonist |
| celiprolol | Antagonist | experimental | Small molecule | ADRB1 antagonist |
| esmolol (brevibloc) | Antagonist | approved | Small molecule | ADRB1 antagonist |
| landiolol | Antagonist | approved | Small molecule | ADRB1 antagonist |
| levobetaxolol (betaxon) | Antagonist | approved | Small molecule | ADRB1 antagonist |
| levobunolol (betagan) | Antagonist | approved | Small molecule | ADRB1 antagonist |
| ly-377604 | Antagonist | experimental | Small molecule | ADRB1 antagonist |
| metipranolol (optipranolol) | Antagonist | approved | Small molecule | ADRB1 antagonist |
| metoprolol (lopressor) | Antagonist | approved | Small molecule | ADRB1 antagonist |
| nadolol (corgard) | Antagonist | approved | Small molecule | ADRB1 antagonist |
| nebivolol (bystolic) | Antagonist | approved | Small molecule | ADRB1 antagonist |
| oxprenolol (trasicor) | Antagonist | approved | Small molecule | ADRB1 antagonist |
| penbutolol (levatol) | Antagonist | approved | Small molecule | ADRB1 antagonist |
| pronetalol | Antagonist | experimental | Small molecule | ADRB1 antagonist |
| propafenone (rythmol) | Antagonist | approved | Small molecule | ADRB1 antagonist |
| propanolol | Antagonist | experimental | Small molecule | ADRB1 antagonist |
| propranolol (inderal) | Antagonist | approved | Small molecule | ADRB1 antagonist |
| sotalol (betapace) | Antagonist | approved | Small molecule | ADRB1 antagonist |
| talinolol | Antagonist | experimental | Small molecule | ADRB1 antagonist |
| timolol (blocadren) | Antagonist | approved | Small molecule | ADRB1 antagonist |
| bevantolol | Inhibitor | experimental | Small molecule | ADRB1 inhibitor |
| cycloprolol | Inhibitor | experimental | Small molecule | ADRB1 inhibitor |
| jnj-54452840 | Inhibitor | experimental | Peptide | ADRB1 inhibitor |
| pindolol (visken) | Partial agonist | approved | Small molecule | ADRB1 partial agonist |
| xamoterol hemifumarate | Partial agonist | experimental | Small molecule | Beta-1 adrenergic receptor partial agonist |