← Mechanisms of action
PGR
SINGLE PROTEINHomo sapiens
Preferred name: Progesterone receptor ChEMBL ↗
Linked proteins
Drugs acting on this target (38)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| cridanimod | Activator | experimental | Small molecule | PGR activator |
| 11 alpha-hydroxyprogesterone | Agonist | experimental | Small molecule | PGR agonist |
| cyproviron | Agonist | experimental | Small molecule | PGR agonist |
| danazol (danocrine) | Agonist | approved | Small molecule | PGR agonist |
| desogestrel (Mercilon) | Agonist | approved | Small molecule | PGR agonist |
| drospirenone (Yasmin) | Agonist | approved | Small molecule | PGR agonist |
| dydrgesterone | Agonist | experimental | Small molecule | PGR agonist |
| dydrogesterone (gynorest) | Agonist | approved | Small molecule | PGR agonist |
| etonogestrel | Agonist | experimental | Small molecule | PGR agonist |
| etynodiol acetate | Agonist | approved | Small molecule | PGR agonist |
| gestodene (Femodene) | Agonist | experimental | Small molecule | PGR agonist |
| hydroxyprogesterone (Delalutin) | Agonist | approved | Small molecule | PGR agonist |
| levonorgestrel | Agonist | experimental | Small molecule | PGR agonist |
| lynestrenol (Exluton) | Agonist | experimental | Small molecule | PGR agonist |
| medroxyprogesterone (provera) | Agonist | approved | Small molecule | PGR agonist |
| megestrol (megace) | Agonist | approved | Small molecule | PGR agonist |
| Nomegestrol acetate | Agonist | experimental | Small molecule | PGR agonist |
| norelgestromin (Evra) | Agonist | approved | Small molecule | PGR agonist |
| norethindrone | Agonist | approved | Small molecule | PGR agonist |
| norethynodrel | Agonist | approved | Small molecule | PGR agonist |
| norgestimate | Agonist | approved | Small molecule | PGR agonist |
| norgestrel (Ovral) | Agonist | approved | Small molecule | PGR agonist |
| orageston | Agonist | experimental | Small molecule | PGR agonist |
| progesterone (progestasert) | Agonist | approved | Small molecule | PGR agonist |
| segesterone (Annovera) | Agonist | approved | Small molecule | PGR agonist |
| trimegestone | Agonist | experimental | Small molecule | PGR agonist |
| lonaprisan | Antagonist | experimental | Small molecule | PGR antagonist |
| mifepristone (mifeprex) | Antagonist | approved | Small molecule | PGR antagonist |
| Norethisterone (norestrone) | Antagonist | experimental | Small molecule | PGR antagonist |
| onapristone | Antagonist | experimental | Small molecule | PGR antagonist |
| pf02413873 | Antagonist | experimental | Small molecule | PGR antagonist |
| way-257027 | Antagonist | experimental | Small molecule | PGR antagonist |
| telepristone | Inhibitor | experimental | Small molecule | PGR inhibitor |
| asoprisnil | Modulator | experimental | Small molecule | PGR modulator |
| chlormadinone | Modulator | experimental | Small molecule | PGR modulator |
| progenta | Modulator | experimental | Small molecule | PGR modulator |
| ulipristal (ella) | Modulator | approved | Small molecule | PGR modulator |
| vilaprisan | Modulator | experimental | Small molecule | PGR modulator |