← Mechanisms of action
CSF1R
SINGLE PROTEINHomo sapiens
Preferred name: Macrophage colony stimulating factor receptor ChEMBL ↗
Linked proteins
Drugs acting on this target (34)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| bc006 | Antagonist | experimental | mAb | csf1r |
| cabiralizumab | Antagonist | experimental | mAb | Macrophage colony stimulating factor receptor antagonist |
| hmpl-653 | Antagonist | experimental | Small molecule | CSF1R |
| abt-869 | Inhibitor | experimental | Small molecule | CSF1R inhibitor |
| amg-820 | Inhibitor | experimental | mAb | CSF1R inhibitor |
| apl-102 | Inhibitor | experimental | Small molecule | CSF1R inhibitor |
| arry-382 | Inhibitor | experimental | Small molecule | CSF1R inhibitor |
| Axatilimab (Niktimvo) | Inhibitor | approved | mAb | Macrophage colony stimulating factor receptor inhibitor |
| c019199 | Inhibitor | experimental | Small molecule | CSF1R inhibitor |
| cabiralizumab | Inhibitor | experimental | mAb | CSF1R inhibitor |
| ei1071 | Inhibitor | experimental | Small molecule | CSF1R inhibitor |
| Elzovantinib | Inhibitor | experimental | Small molecule | CSF1R inhibitor |
| emactuzumab | Inhibitor | experimental | mAb | CSF1R inhibitor |
| enmd 2076 | Inhibitor | experimental | Small molecule | CSF1R inhibitor |
| imc-cs4 | Inhibitor | experimental | mAb | CSF1R inhibitor |
| jnj-40346527 | Inhibitor | experimental | Small molecule | CSF1R inhibitor |
| ly3022855 | Inhibitor | experimental | mAb | CSF1R inhibitor |
| nindetanib | Inhibitor | experimental | Small molecule | CSF1R inhibitor |
| nms-03592088 | Inhibitor | experimental | Small molecule | CSF1R inhibitor |
| pazopanib (votrient) | Inhibitor | approved | Small molecule | CSF1R inhibitor |
| pexidartinib (Turalio) | Inhibitor | approved | Small molecule | CSF1R inhibitor |
| plx-5622 | Inhibitor | experimental | Small molecule | CSF1R inhibitor |
| plx-7486 | Inhibitor | experimental | Small molecule | CSF1R inhibitor |
| plx73086 | Inhibitor | experimental | Small molecule | CSF1R inhibitor |
| prv-6527 | Inhibitor | experimental | Small molecule | CSF1R inhibitor |
| q702 | Inhibitor | experimental | Small molecule | CSF1R inhibitor |
| quizartinib (VANFLYTA) | Inhibitor | approved | Small molecule | CSF1R inhibitor |
| sb1578 | Inhibitor | experimental | Small molecule | CSF1R inhibitor |
| Seralutinib | Inhibitor | experimental | Small molecule | Macrophage colony stimulating factor receptor inhibitor |
| sunitinib (sutent) | Inhibitor | approved | Small molecule | CSF1R inhibitor |
| syha1813 | Inhibitor | experimental | Small molecule | CSF1R inhibitor |
| vatalanib | Inhibitor | experimental | Small molecule | CSF1R inhibitor |
| vimseltinib | Inhibitor | approved | Small molecule | CSF1R inhibitor |
| [11c]cppc | Radiopharmaceutical | experimental | Small molecule | CSF1R radiopharmaceutical |