← Mechanisms of action
HTR4
SINGLE PROTEINHomo sapiens
Preferred name: Serotonin 4 (5-HT4) receptor ChEMBL ↗
Linked proteins
Drugs acting on this target (32)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| mescaline | Activator | experimental | Small molecule | HTR4 activator |
| prucalopride succinate (Motegrity) | Activator | approved | Small molecule | HTR4 activator |
| cinitapride | Agonist | experimental | Small molecule | HTR4 agonist |
| cisapride (Propulsid) | Agonist | approved | Small molecule | HTR4 agonist |
| clebopride maleate | Agonist | experimental | Small molecule | HTR4 agonist |
| da-6886 | Agonist | experimental | Small molecule | HTR4 agonist |
| levosulpiride | Agonist | experimental | Small molecule | Serotonin 4 (5-HT4) receptor agonist |
| m-chlorophenylpiperazine | Agonist | experimental | Small molecule | HTR4 agonist |
| metoclopramide (reglan) | Agonist | approved | Small molecule | HTR4 agonist |
| mosapride | Agonist | experimental | Small molecule | HTR4 agonist |
| naronapride | Agonist | experimental | Small molecule | HTR4 agonist |
| pf-00885706 | Agonist | experimental | Small molecule | HTR4 agonist |
| pf-04995274 | Agonist | experimental | Small molecule | HTR4 agonist |
| prucalopride succinate (Motegrity) | Agonist | approved | Small molecule | Serotonin 4 (5-HT4) receptor agonist |
| relenopride | Agonist | experimental | Small molecule | HTR4 agonist |
| renzapride | Agonist | experimental | Small molecule | HTR4 agonist |
| revexepride | Agonist | experimental | Small molecule | HTR4 agonist |
| serotonin | Agonist | experimental | Small molecule | HTR4 agonist |
| tak-951 | Agonist | experimental | Peptide | HTR4 agonist |
| tak-954 | Agonist | experimental | Small molecule | HTR4 agonist |
| td-8954 | Agonist | experimental | Small molecule | HTR4 agonist |
| velusetrag | Agonist | experimental | Small molecule | HTR4 agonist |
| pcs12852 | Antagonist | experimental | Small molecule | HTR4 antagonist |
| piboserod | Antagonist | experimental | Small molecule | HTR4 antagonist |
| escalitopram (Lexapro) | Inhibitor | experimental | Small molecule | HTR4 inhibitor |
| jx11502ma | Inhibitor | experimental | Small molecule | HTR4 inhibitor |
| capeserod | Partial agonist | experimental | Small molecule | HTR4 partial agonist |
| pf-03382792 | Partial agonist | experimental | Small molecule | HTR4 partial agonist |
| prx-03140 | Partial agonist | experimental | Small molecule | HTR4 partial agonist |
| rq-00000010 | Partial agonist | experimental | Small molecule | HTR4 partial agonist |
| tegaserod (zelnorm) | Partial agonist | approved | Small molecule | HTR4 partial agonist |
| Usmarapride | Partial agonist | experimental | Small molecule | HTR4 partial agonist |