← Mechanisms of action
Pyruvate dehydrogenase kinase
PROTEIN FAMILYHomo sapiens
Linked proteins
- [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 2, mitochondrial (PDK2) ↗
- [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 3, mitochondrial (PDK3) ↗
- [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial (PDK4) ↗
- [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial (PDK1) ↗
Drugs acting on this target (4)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| arsenic | Inhibitor | experimental | Small molecule | Pyruvate dehydrogenase kinase inhibitor |
| cpi 613 | Inhibitor | experimental | Small molecule | Pyruvate dehydrogenase kinase inhibitor |
| devimistat | Inhibitor | experimental | Small molecule | Pyruvate dehydrogenase kinase inhibitor |
| sodium dichloroacetate | Inhibitor | experimental | Small molecule | Pyruvate dehydrogenase kinase inhibitor |