← Mechanisms of action
Neuronal acetylcholine receptor; alpha4/beta2
PROTEIN COMPLEXHomo sapiens
Linked proteins
Drugs acting on this target (14)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| azd-1446 | Agonist | experimental | Small molecule | Neuronal acetylcholine receptor; alpha4/beta2 agonist |
| nicotine (nicorette) | Agonist | approved | Small molecule | Neuronal acetylcholine receptor; alpha4/beta2 agonist |
| sofinicline | Agonist | experimental | Small molecule | Neuronal acetylcholine receptor; alpha4/beta2 agonist |
| tc-6499 | Agonist | experimental | Small molecule | Neuronal acetylcholine receptor; alpha4/beta2 agonist |
| varenicline (chantix) | Agonist | approved | Small molecule | Neuronal acetylcholine receptor; alpha4/beta2 agonist |
| dexmecamylamine | Antagonist | experimental | Small molecule | Neuronal acetylcholine receptor; alpha4/beta2 antagonist |
| tc-2216 | Antagonist | experimental | Small molecule | Neuronal acetylcholine receptor; alpha4/beta2 antagonist |
| Ropanicant | Inhibitor | experimental | Small molecule | Neuronal acetylcholine receptor; alpha4/beta2 inhibitor |
| azd-3480 | Partial agonist | experimental | Small molecule | Neuronal acetylcholine receptor; alpha4/beta2 partial agonist |
| cp-601927 | Partial agonist | experimental | Small molecule | Neuronal acetylcholine receptor; alpha4/beta2 partial agonist |
| cytisinicline | Partial agonist | experimental | Small molecule | Neuronal acetylcholine receptor; alpha4/beta2 partial agonist |
| dianicline | Partial agonist | experimental | Small molecule | Neuronal acetylcholine receptor; alpha4/beta2 partial agonist |
| gts-21 | Partial agonist | experimental | Small molecule | Neuronal acetylcholine receptor; alpha4/beta2 partial agonist |
| varenicline (chantix) | Partial agonist | approved | Small molecule | Neuronal acetylcholine receptor; alpha4/beta2 partial agonist |