← Mechanisms of action
ALK
SINGLE PROTEINHomo sapiens
Preferred name: ALK tyrosine kinase receptor ChEMBL ↗
Linked proteins
Drugs acting on this target (31)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| ds-6016a | Antagonist | experimental | mAb | ALK antagonist |
| entrectinib (Rozlytrek) | Antagonist | approved | Small molecule | ALK antagonist |
| lorlatinib (lorbrena) | Antagonist | approved | Small molecule | ALK antagonist |
| nvl-655 | Antagonist | experimental | Small molecule | ALK |
| sy-3505 | Antagonist | experimental | Small molecule | ALK |
| tgrx-326 | Antagonist | experimental | Small molecule | alk |
| autologous halk.car t cells | Immunity, passive | experimental | Cell therapy | ALK immunity, passive |
| alectinib (alecensa) | Inhibitor | approved | Small molecule | ALK inhibitor |
| alk202 | Inhibitor | experimental | mAb | ALK inhibitor |
| alkotinib | Inhibitor | experimental | Small molecule | ALK inhibitor |
| apg-2449 | Inhibitor | experimental | Small molecule | ALK inhibitor |
| asp-3026 | Inhibitor | experimental | Small molecule | ALK inhibitor |
| brigatinib (alunbrig) | Inhibitor | approved | Small molecule | ALK inhibitor |
| cep-37440 | Inhibitor | experimental | Small molecule | ALK inhibitor |
| ceritinib (zykadia) | Inhibitor | approved | Small molecule | ALK inhibitor |
| crizotinib (xalkori) | Inhibitor | approved | Small molecule | ALK inhibitor |
| ensartinib (Ensacove) | Inhibitor | approved | Small molecule | ALK inhibitor |
| entrectinib (Rozlytrek) | Inhibitor | approved | Small molecule | ALK tyrosine kinase receptor inhibitor |
| fn-1501 | Inhibitor | experimental | Small molecule | ALK inhibitor |
| imm47 | Inhibitor | experimental | mAb | ALK inhibitor |
| Iruplinalkib | Inhibitor | experimental | Small molecule | ALK inhibitor |
| lorlatinib (lorbrena) | Inhibitor | approved | Small molecule | ALK tyrosine kinase receptor inhibitor |
| plb1003 | Inhibitor | experimental | Small molecule | ALK inhibitor |
| repotrectinib (Augtyro) | Inhibitor | approved | Small molecule | ALK inhibitor |
| saf-189s | Inhibitor | experimental | Small molecule | ALK inhibitor |
| sim1803-1a | Inhibitor | experimental | Small molecule | ALK inhibitor |
| tpx-0131 | Inhibitor | experimental | Small molecule | ALK inhibitor |
| tq-b3101 | Inhibitor | experimental | Small molecule | ALK inhibitor |
| tsr-011 | Inhibitor | experimental | Small molecule | ALK inhibitor |
| ty-2136b | Inhibitor | experimental | Small molecule | ALK inhibitor |
| xzp-3621 | Inhibitor | experimental | Small molecule | ALK inhibitor |