← Mechanisms of action
EML4-ALK
CHIMERIC PROTEINHomo sapiens
Linked proteins
Drugs acting on this target (5)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| alectinib (alecensa) | Inhibitor | approved | Small molecule | EML4-ALK |
| ceritinib (zykadia) | Inhibitor | approved | Small molecule | EML4-ALK |
| crizotinib (xalkori) | Inhibitor | approved | Small molecule | EML4-ALK |
| lorlatinib (lorbrena) | Inhibitor | approved | Small molecule | EML4-ALK inhibitor |
| plb1003 | Inhibitor | experimental | Small molecule | EML4-ALK inhibitor |