← Mechanisms of action
EDNRA
SINGLE PROTEINHomo sapiens
Preferred name: Endothelin receptor ET-A ChEMBL ↗
Linked proteins
Drugs acting on this target (14)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| atrasentan hydrochloride | Antagonist | approved | Small molecule | EDNRA antagonist |
| Avosentan | Antagonist | experimental | Small molecule | EDNRA antagonist |
| bq-123 | Antagonist | experimental | Peptide | Endothelin receptor ET-A antagonist |
| clazosentan | Antagonist | experimental | Small molecule | EDNRA antagonist |
| darusentan | Antagonist | experimental | Small molecule | EDNRA antagonist |
| enrasentan | Antagonist | experimental | Small molecule | EDNRA antagonist |
| nebentan | Antagonist | experimental | Small molecule | EDNRA antagonist |
| sc0062 | Antagonist | experimental | Small molecule | EDNRA antagonist |
| sitaxentan | Antagonist | experimental | Small molecule | EDNRA antagonist |
| sparsentan (FILSPARI) | Antagonist | approved | Small molecule | EDNRA antagonist |
| tezosentan | Antagonist | experimental | Small molecule | EDNRA antagonist |
| zibotentan | Antagonist | experimental | Small molecule | EDNRA antagonist |
| Avosentan | Inhibitor | experimental | Small molecule | EDNRA inhibitor |
| per-001 | Inhibitor | experimental | Small molecule | EDNRA inhibitor |