← Mechanisms of action
Q72547
SINGLE PROTEINHuman immunodeficiency virus 1
Preferred name: Human immunodeficiency virus type 1 reverse transcriptase ChEMBL ↗
Linked proteins
Drugs acting on this target (29)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| doravirine (pifeltro) | Antagonist | approved | Small molecule | Q72547 antagonist |
| abacavir (ziagen) | Inhibitor | approved | Small molecule | Q72547 inhibitor |
| amdoxovir | Inhibitor | experimental | Small molecule | Human immunodeficiency virus type 1 reverse transcriptase inhibitor |
| apricitabine | Inhibitor | experimental | Small molecule | Human immunodeficiency virus type 1 reverse transcriptase inhibitor |
| atevirdine | Inhibitor | experimental | Small molecule | Human immunodeficiency virus type 1 reverse transcriptase inhibitor |
| capravirine | Inhibitor | experimental | Small molecule | Human immunodeficiency virus type 1 reverse transcriptase inhibitor |
| censavudine | Inhibitor | experimental | Small molecule | Human immunodeficiency virus type 1 reverse transcriptase inhibitor |
| dapivirine | Inhibitor | experimental | Small molecule | Reverse transcriptase inhibitor |
| delavirdine (rescriptor) | Inhibitor | approved | Small molecule | Q72547 inhibitor |
| dexelvucitabine | Inhibitor | experimental | Small molecule | Human immunodeficiency virus type 1 reverse transcriptase inhibitor |
| didanosine (videx) | Inhibitor | approved | Small molecule | Q72547 inhibitor |
| efavirenz (sustiva) | Inhibitor | approved | Small molecule | Q72547 inhibitor |
| elvucitabine | Inhibitor | experimental | Small molecule | Human immunodeficiency virus type 1 reverse transcriptase inhibitor |
| emivirine | Inhibitor | experimental | Small molecule | Human immunodeficiency virus type 1 reverse transcriptase inhibitor |
| emtricitabine (emtriva) | Inhibitor | approved | Small molecule | Q72547 inhibitor |
| etravirine (intelence) | Inhibitor | approved | Small molecule | Q72547 inhibitor |
| islatravir | Inhibitor | experimental | Small molecule | Human immunodeficiency virus type 1 reverse transcriptase inhibitor |
| lamivudine (epivir) | Inhibitor | approved | Small molecule | Q72547 inhibitor |
| lersivirine | Inhibitor | experimental | Small molecule | Human immunodeficiency virus type 1 reverse transcriptase inhibitor |
| nevirapine (viramune) | Inhibitor | approved | Small molecule | Q72547 inhibitor |
| rilpivirine (edurant) | Inhibitor | approved | Small molecule | Q72547 inhibitor |
| Rovafovir etalafenamide | Inhibitor | experimental | Small molecule | Human immunodeficiency virus type 1 reverse transcriptase inhibitor |
| stavudine (zerit) | Inhibitor | approved | Small molecule | Q72547 inhibitor |
| tenofovir (viread) | Inhibitor | approved | Small molecule | Q72547 inhibitor |
| tenofovir alafenamide (genvoya) | Inhibitor | approved | Small molecule | Q72547 inhibitor |
| Tenofovir exalidex | Inhibitor | experimental | Small molecule | Human immunodeficiency virus type 1 reverse transcriptase inhibitor |
| zalcitabine (hivid) | Inhibitor | approved | Small molecule | Q72547 inhibitor |
| zidovudine (retrovir) | Inhibitor | approved | Small molecule | Q72547 inhibitor |
| doravirine (pifeltro) | Negative allosteric modulator | approved | Small molecule | Reverse transcriptase negative allosteric modulator |