← Mechanisms of action
FLT3
SINGLE PROTEINHomo sapiens
Preferred name: Tyrosine-protein kinase receptor FLT3 ChEMBL ↗
Linked proteins
Drugs acting on this target (46)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| cdx-301 | Agonist | experimental | Recombinant protein | Tyrosine-protein kinase receptor FLT3 agonist |
| stk1-ligand | Agonist | experimental | Recombinant protein | FLT3 agonist |
| cln-049 | Binding agent | experimental | mAb | FLT3 |
| 4sc-203 | Inhibitor | experimental | Small molecule | FLT3 inhibitor |
| abt-869 | Inhibitor | experimental | Small molecule | FLT3 inhibitor |
| ags62p1 | Inhibitor | experimental | mAb | FLT3 inhibitor |
| akn-028 | Inhibitor | experimental | Small molecule | FLT3 inhibitor |
| amg 427 | Inhibitor | experimental | mAb | FLT3 inhibitor |
| amuvatinib | Inhibitor | experimental | Small molecule | FLT3 inhibitor |
| as-602868 | Inhibitor | experimental | Small molecule | FLT3 inhibitor |
| at9283 | Inhibitor | experimental | Small molecule | FLT3 inhibitor |
| cep2563 | Inhibitor | experimental | Small molecule | FLT3 inhibitor |
| clifutinib | Inhibitor | experimental | Small molecule | FLT3 inhibitor |
| cm-082 | Inhibitor | experimental | Small molecule | FLT3 inhibitor |
| crenolanib | Inhibitor | experimental | Small molecule | FLT3 inhibitor |
| enmd 2076 | Inhibitor | experimental | Small molecule | FLT3 inhibitor |
| famitinib | Inhibitor | experimental | Small molecule | FLT3 inhibitor |
| fedratinib (Inrebic) | Inhibitor | approved | Small molecule | FLT3 inhibitor |
| flysyn | Inhibitor | experimental | mAb | Tyrosine-protein kinase receptor FLT3 inhibitor |
| foretinib | Inhibitor | experimental | Small molecule | FLT3 inhibitor |
| gb3226 | Inhibitor | experimental | Small molecule | FLT3 inhibitor |
| gilteritinib | Inhibitor | approved | Small molecule | FLT3 inhibitor |
| hpb-092 | Inhibitor | experimental | Small molecule | FLT3 inhibitor |
| imc-eb10 | Inhibitor | experimental | mAb | FLT3 inhibitor |
| kw2449 | Inhibitor | experimental | Small molecule | FLT3 inhibitor |
| lestaurtinib | Inhibitor | experimental | Small molecule | FLT3 inhibitor |
| lomonitinib | Inhibitor | experimental | Small molecule | FLT3 inhibitor |
| midostaurin (rydapt) | Inhibitor | approved | Small molecule | FLT3 inhibitor |
| nindetanib | Inhibitor | experimental | Small molecule | FLT3 inhibitor |
| ningetinib | Inhibitor | experimental | Small molecule | Tyrosine-protein kinase receptor FLT3 inhibitor |
| nsc-645809 | Inhibitor | experimental | Small molecule | FLT3 inhibitor |
| nvp-ast487 | Inhibitor | experimental | Small molecule | FLT3 inhibitor |
| pacritinib (Vonjo) | Inhibitor | approved | Small molecule | FLT3 inhibitor |
| pexidartinib (Turalio) | Inhibitor | approved | Small molecule | FLT3 inhibitor |
| progenipoietin | Inhibitor | experimental | Recombinant protein | FLT3 inhibitor |
| quizartinib (VANFLYTA) | Inhibitor | approved | Small molecule | FLT3 inhibitor |
| rg1530 | Inhibitor | experimental | Small molecule | FLT3 inhibitor |
| sb1578 | Inhibitor | experimental | Small molecule | FLT3 inhibitor |
| sklb1028 | Inhibitor | experimental | Small molecule | FLT3 inhibitor |
| sorafenib (nexavar) | Inhibitor | approved | Small molecule | FLT3 inhibitor |
| su14813 | Inhibitor | experimental | Small molecule | FLT3 inhibitor |
| sunitinib (sutent) | Inhibitor | approved | Small molecule | FLT3 inhibitor |
| tandutinib | Inhibitor | experimental | Small molecule | FLT3 inhibitor |
| tg02 | Inhibitor | experimental | Small molecule | FLT3 inhibitor |
| tt-00973 | Inhibitor | experimental | Small molecule | FLT3 inhibitor |
| xl999 | Inhibitor | experimental | Small molecule | FLT3 inhibitor |