← Mechanisms of action

CDK2

SINGLE PROTEINHomo sapiens
Preferred name: Cyclin-dependent kinase 2 ChEMBL ↗

Linked proteins

Drugs acting on this target (26)

Active Pharmaceutical Ingredient Mechanism Type Approval Status API Type Mechanism of Action
blu-222AntagonistexperimentalSmall moleculeCDK2
bg-75098DegraderexperimentalSmall moleculeCDK2 degrader
nkt3964DegraderexperimentalSmall moleculeCDK2 degrader
nkt5097DegraderexperimentalSmall moleculeCDK2 degrader
7-hydroxystaurosporineInhibitorexperimentalSmall moleculeCDK2 inhibitor
ag-24322InhibitorexperimentalSmall moleculeCDK2 inhibitor
alvocidibInhibitorexperimentalSmall moleculeCDK2 inhibitor
arts-011InhibitorexperimentalSmall moleculeCDK2 inhibitor
avzo-021InhibitorexperimentalSmall moleculeCDK2 inhibitor
azd8421InhibitorexperimentalSmall moleculeCDK2 inhibitor
bg-68501InhibitorexperimentalSmall moleculeCDK2 inhibitor
bms 387032InhibitorexperimentalSmall moleculeCDK2 inhibitor
dinaciclibInhibitorexperimentalSmall moleculeCDK2 inhibitor
gdc-4198InhibitorexperimentalSmall moleculeCDK2 inhibitor
hrs-3802InhibitorexperimentalSmall moleculeCDK2 inhibitor
incb123667InhibitorexperimentalSmall moleculeCDK2 inhibitor
indirubin sulfateInhibitorexperimentalSmall moleculeCDK2 inhibitor
milciclibInhibitorexperimentalSmall moleculeCDK2 inhibitor
nkt3447InhibitorexperimentalSmall moleculeCDK2 inhibitor
pf-07104091InhibitorexperimentalSmall moleculeCDK2 inhibitor
rg547InhibitorexperimentalSmall moleculeCDK2 inhibitor
rgb286638InhibitorexperimentalSmall moleculeCDK2 inhibitor
rgt-419bInhibitorexperimentalSmall moleculeCDK2 inhibitor
roscovitineInhibitorexperimentalSmall moleculeCDK2 inhibitor
tg02InhibitorexperimentalSmall moleculeCDK2 inhibitor
tyk-00540InhibitorexperimentalSmall moleculeCDK2 inhibitor