← Mechanisms of action

CDK2/CDK4

PROTEIN FAMILYHomo sapiens

Linked proteins

Drugs acting on this target (8)

Active Pharmaceutical Ingredient Mechanism Type Approval Status API Type Mechanism of Action
trilaciclib (Cosela)AntagonistapprovedSmall moleculeCDK2/CDK4 antagonist
arts-021InhibitorexperimentalSmall moleculeCDK2/CDK4 inhibitor
cyc065InhibitorexperimentalSmall moleculeCDK2/CDK4 inhibitor
incb0123667InhibitorexperimentalSmall moleculeCDK2/CDK4 inhibitor
inx-315InhibitorexperimentalSmall moleculeCDK2/CDK4 inhibitor
nuv-422InhibitorexperimentalSmall moleculeCDK2/CDK4 inhibitor
pf-06873600InhibitorexperimentalSmall moleculeCDK2/CDK4 inhibitor
syh2043InhibitorexperimentalSmall moleculeCDK2/CDK4 inhibitor