← Mechanisms of action
DPP4
SINGLE PROTEINHomo sapiens
Preferred name: Dipeptidyl peptidase IV ChEMBL ↗
Linked proteins
Drugs acting on this target (34)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| alogliptin (nesina) | Inhibitor | approved | Small molecule | DPP4 inhibitor |
| anagliptin | Inhibitor | experimental | Small molecule | Dipeptidyl peptidase IV inhibitor |
| begelomab | Inhibitor | experimental | mAb | DPP4 inhibitor |
| bi 14332 | Inhibitor | experimental | Small molecule | DPP4 inhibitor |
| Bisegliptin | Inhibitor | experimental | Small molecule | Dipeptidyl peptidase IV inhibitor |
| bms-767778 | Inhibitor | experimental | Small molecule | DPP4 inhibitor |
| carmegliptin | Inhibitor | experimental | Small molecule | DPP4 inhibitor |
| cofrogliptin | Inhibitor | experimental | Small molecule | DPP4 inhibitor |
| cpl-2009-0031 | Inhibitor | experimental | Small molecule | DPP4 inhibitor |
| denagliptin | Inhibitor | experimental | Small molecule | DPP4 inhibitor |
| dutogliptin | Inhibitor | experimental | Small molecule | DPP4 inhibitor |
| evogliptin (Suganon) | Inhibitor | experimental | Small molecule | Dipeptidyl peptidase IV inhibitor |
| gemigliptin (Zemiglo) | Inhibitor | experimental | Small molecule | DPP4 inhibitor |
| glimepiride (amaryl) | Inhibitor | approved | Small molecule | DPP4 inhibitor |
| gosogliptin | Inhibitor | experimental | Small molecule | DPP4 inhibitor |
| grc 8200 | Inhibitor | experimental | Small molecule | DPP4 inhibitor |
| ip10.c8 | Inhibitor | experimental | Small molecule | DPP4 inhibitor |
| linagliptin (tradjenta) | Inhibitor | approved | Small molecule | DPP4 inhibitor |
| omarigliptin | Inhibitor | experimental | Small molecule | DPP4 inhibitor |
| prusogliptin | Inhibitor | experimental | Small molecule | DPP4 inhibitor |
| Retagliptin | Inhibitor | experimental | Small molecule | DPP4 inhibitor |
| saxagliptin (onglyza) | Inhibitor | approved | Small molecule | DPP4 inhibitor |
| sdp-4 | Inhibitor | experimental | Small molecule | DPP4 inhibitor |
| shr117887 | Inhibitor | experimental | Small molecule | DPP4 inhibitor |
| sitagliptin (januvia) | Inhibitor | approved | Small molecule | DPP4 inhibitor |
| sk-0403 | Inhibitor | experimental | Small molecule | DPP4 inhibitor |
| syr-619 | Inhibitor | experimental | Small molecule | DPP4 inhibitor |
| talabostat | Inhibitor | experimental | Small molecule | DPP4 inhibitor |
| teneligliptin (Tenelia) | Inhibitor | experimental | Small molecule | DPP4 inhibitor |
| tq-f3083 | Inhibitor | experimental | Small molecule | DPP4 inhibitor |
| trelagliptin | Inhibitor | experimental | Small molecule | DPP4 inhibitor |
| vildagliptin | Inhibitor | experimental | Small molecule | DPP4 inhibitor |
| ys110 | Inhibitor | experimental | mAb | DPP4 inhibitor |
| zydpla1 | Inhibitor | experimental | Small molecule | DPP4 inhibitor |