deslorelin
Animal productexperimental
Deslorelin, sold under the brand name Suprelorin among others, is an injectable gonadotropin releasing hormone superagonist which is used in veterinary medicine for various indications. — Wikipedia
Clinical trial activity
4 trials · 3 clinical orgs · 0 marketing orgs
Phase 1
1
Phase 2
3
Phase 3
0
Phase 4
0
Earliest trial started Nov 1, 1983 (NCT00001190)
Timeline
Indications
Mechanism of action
GNRHR agonist
Chemistry & pharmacology
Loading structure…
SMILES
CCNC(=O)[C@@H]1CCCN1C(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@H](CO)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@H](Cc1c[nH]cn1)NC(=O)[C@@H]1CCC(=O)N1- Mol. weight
- 1282.47 g/mol
- Chirality
- Single Stereoisomer
- Inorganic
- No
- Polymer
- No
Oral
No
Parenteral
No
Topical
No
Sources
- WikipediaDeslorelin ↗
- ChEMBLCHEMBL2365665 ↗
Also known as
- 6-trp-10-n-et-glynh2-lhrh
- deslorelin
- deslorelin
- deslorelin
- deslorelin
- deslorelin acetate
- d-trp(6)-n-et-d-glynh2(10)-lhrh
- d-trp lhrh-pea
- d-trp lhrh-pea
- gnrh, trp(6)-n-et-glynh2(10)-
- lhrh, trp(6)-n-et-glynh2(10)-
- lhrh, tryptophyl(6)-n-ethylglycinamide(10)-
- ovuplant
- somagard
- somagard [as acetate]
Clinical trials
| NCT ID | Phase | Start date | Sponsor(s) |
|---|---|---|---|
| NCT00080756 | Phase 2 | Feb 1, 2004 | City of Hope National Medical Center, National Cancer Institute (NCI) |
| NCT00001521 | Phase 1 | Feb 2, 1996 | National Institutes of Health (NIH) |
| NCT00001202 | Phase 2 | Jan 1, 1985 | National Institutes of Health (NIH) |
| NCT00001190 | Phase 2 | Nov 1, 1983 | National Institutes of Health (NIH) |
Showing 4 of 4 trials
Page 1 / 1
Organizations
Research & Development (3)
| Organization | Org type | Trials | As lead sponsor | Phases | Earliest year |
|---|---|---|---|---|---|
| National Institutes of Health (NIH) | Government | 3 | 3 | 2 | 1983 |
| City of Hope National Medical Center | Academic/Hospital | 1 | 1 | 1 | 2004 |
| National Cancer Institute (NCI) | Government | 1 | 0 | 1 | 2004 |
3 organizations
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