← Mechanisms of action
GNRHR
SINGLE PROTEINHomo sapiens
Preferred name: Gonadotropin-releasing hormone receptor ChEMBL ↗
Linked proteins
Drugs acting on this target (35)
| Active Pharmaceutical Ingredient | Mechanism Type ▲ | Approval Status | API Type | Mechanism of Action |
|---|---|---|---|---|
| buserelin (receptal) | Agonist | experimental | Small molecule | GNRHR agonist |
| debio 4326 | Agonist | experimental | Small molecule | GNRHR agonist |
| deslorelin | Agonist | experimental | Animal product | GNRHR agonist |
| follitropin alfa (Gonal-F) | Agonist | approved | Recombinant protein | GNRHR agonist |
| gonadorelin (factrel) | Agonist | approved | Small molecule | GNRHR agonist |
| Gonadotropin-releasing hormone | Agonist | experimental | Small molecule | GNRHR agonist |
| goserelin (zoladex) | Agonist | approved | Small molecule | GNRHR agonist |
| histrelin (supprelin) | Agonist | approved | Small molecule | GNRHR agonist |
| leuprolide (lupron) | Agonist | approved | Small molecule | GNRHR agonist |
| nafarelin (synarel) | Agonist | approved | Small molecule | GNRHR agonist |
| triptorelin (Trelstar) | Agonist | approved | Peptide | GNRHR agonist |
| zoptarelin doxorubicin | Agonist | experimental | Small molecule | GNRHR agonist |
| abarelix (plenaxis) | Antagonist | approved | Small molecule | GNRHR antagonist |
| acyline | Antagonist | experimental | Small molecule | Gonadotropin-releasing hormone receptor antagonist |
| bay1214784 | Antagonist | experimental | Small molecule | GNRHR antagonist |
| cetrorelix (cetrotide) | Antagonist | approved | Small molecule | GNRHR antagonist |
| degarelix acetate (firmagon) | Antagonist | approved | Peptide | GNRHR antagonist |
| dw4902 | Antagonist | experimental | Small molecule | GNRHR antagonist |
| elagolix (orilissa) | Antagonist | approved | Small molecule | GNRHR antagonist |
| ganirelix | Antagonist | approved | Peptide | GNRHR antagonist |
| klh-2109 | Antagonist | experimental | Small molecule | GNRHR antagonist |
| linzagolix | Antagonist | experimental | Small molecule | Gonadotropin-releasing hormone receptor antagonist |
| Opigolix | Antagonist | experimental | Small molecule | GNRHR antagonist |
| ozarelix | Antagonist | experimental | Peptide | GNRHR antagonist |
| relugolix (ORGOVYX) | Antagonist | approved | Small molecule | GNRHR antagonist |
| ski2670 | Antagonist | experimental | Small molecule | GNRHR antagonist |
| sufugolix | Antagonist | experimental | Small molecule | GNRHR antagonist |
| teverelix | Antagonist | experimental | Small molecule | GNRHR antagonist |
| tu2670 | Antagonist | experimental | Small molecule | GNRHR antagonist |
| tu7710 | Antagonist | experimental | Small molecule | GNRHR antagonist |
| veru-100 | Antagonist | experimental | Peptide | GNRHR antagonist |
| acyline | Inhibitor | experimental | Small molecule | GNRHR inhibitor |
| askc202 | Inhibitor | experimental | Small molecule | GNRHR inhibitor |
| linzagolix | Inhibitor | experimental | Small molecule | GNRHR inhibitor |
| shr7280 | Inhibitor | experimental | Small molecule | GNRHR inhibitor |