tricaprylyl glycerol

Small moleculeexperimental

Clinical trial activity

18 trials · 11 clinical orgs · 0 marketing orgs

Phase 1
10
Phase 2
3
Phase 3
3
Phase 4
1

Earliest trial started Sep 24, 2010 (NCT01211782)

Timeline

2010s

  1. Jan 1, 2010

    Earliest Phase 2 Sponsor(trial)

  2. Jan 1, 2015

    Earliest Phase 1 Sponsor(trial)

2020s

  1. Jan 1, 2020

    Earliest Phase 3 Sponsor(trial)

Indications

Approved for

Mechanism of action

Chemistry & pharmacology

Loading structure…

SMILES

CCCCCCCC(=O)OCC(COC(=O)CCCCCCC)OC(=O)CCCCCCC
Mol. weight
470.69 g/mol
Lipinski Ro5
1 violation(s)
Rule of 3
No
Chirality
Achiral Molecule
Inorganic
No
Polymer
No

Oral

No

Parenteral

No

Topical

No

Sources

Also known as

  • ac-sd-01
  • caprylic acid triglyceride
  • caprylic acid triglyceride
  • caprylic triglyceride
  • caprylic triglyceride
  • caprylic triglyceride
  • caprylidene
  • caprylidene
  • glycerol tricaprylate
  • glycerol tricaprylate
  • glycerol trioctanoate
  • glycerol trioctanoate
  • glyceryl tricaprylate
  • glyceryl trioctanoate
  • octanoic acid, 1,2,3- propanetriyl ester
  • panasate 800
  • tricaprilin
  • tricaprilin
  • tricaprylin
  • tricaprylin
  • tricaprylin
  • tricaprylyl glycerin
  • tricaprylyl glycerin
  • tricaprylyl glycerol
  • tricaprylyl glycerol
  • trioctanoin
  • trioctanoin
  • trioctanoin
  • trioctanoylglyceride

Clinical trials

NCT IDPhaseStart dateSponsor(s)
NCT05809908Phase 3Jan 31, 2024Cerecin
NCT04727970Phase 1Nov 30, 2021Cerecin
NCT05028114Phase 1Aug 31, 2021Cerecin
NCT04437199Phase 2Aug 27, 2020Cerecin
NCT04187547Phase 3Apr 30, 2020Cerecin
NCT04268953Phase 1Feb 28, 2020Cerecin
NCT03971123Phase 1Aug 6, 2019Cerecin
NCT03628352Phase 1Sep 10, 2018Cerecin, Senopsys, LLC
NCT03551769Phase 1Aug 5, 2018Cerecin
NCT03223389N/AAug 7, 2017University of Copenhagen
NCT03063645Phase 1Mar 11, 2017Celerion, Cerecin
NCT02833012Phase 1Jul 1, 2016Celerion, Cerecin
NCT02747602Phase 1Apr 1, 2016Celerion, Cerecin
NCT02602158Early Phase 1 (Phase 1)Oct 1, 2015University of Zurich
NCT02679222N/AJun 30, 2015University of Sherbrooke
NCT01848327N/AFeb 1, 2013Cerecin, National Multiple Sclerosis Society, University of Miami
NCT01122329Phase 4Oct 1, 2010John Douglas French Foundation, University of California, Los Angeles
NCT01211782Phase 2/Phase 3 (Phase 3)Sep 24, 2010Cerecin, Meridien Research
Showing 18 of 18 trials
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Organizations

Research & Development (11)

OrganizationOrg typeTrialsAs lead sponsorPhasesEarliest year
CerecinFor profit141342010
CelerionFor profit3012016
John Douglas French FoundationAcademic/Hospital1012010
Meridien ResearchFor profit1012010
National Multiple Sclerosis SocietyAcademic/Hospital1012013
Senopsys, LLCFor profit1012018
University of California, Los AngelesAcademic/Hospital1112010
University of CopenhagenAcademic/Hospital1112017
University of MiamiAcademic/Hospital1112013
University of SherbrookeAcademic/Hospital1112015
University of ZurichAcademic/Hospital1112015
11 organizations
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