levonordefrin

Trade name: Neo-Cobefrine

Small moleculeapproved

Approved

Sep 19, 1952

Levonordefrin acts as a topical nasal decongestant and vasoconstrictor, most often used in dentistry. It is administered in a pre-mixed solution with local anesthetics, such as mepivacaine or procaine. — NCATS

Clinical trial activity

3 trials · 2 clinical orgs · 6 marketing orgs

Phase 1
0
Phase 2
1
Phase 3
1
Phase 4
0

Earliest trial started Oct 22, 2020 (NCT04561921)

Timeline

1950s

  1. Sep 19, 1952

    Kodak — Earliest FDA Approval

  2. Sep 19, 1952

    Kodak — NDA Organization

1960s

  1. Jan 6, 1960

    Kodak — NDA Secondary Org

1970s

  1. Jan 22, 1976

    Belmora — Marketing Organization

  2. Feb 6, 1976

    Septodont — Marketing Organization

  3. Apr 15, 1976

    Solvay — Marketing Organization

1980s

  1. Oct 10, 1984

    Deproco — Marketing Organization

  2. Apr 14, 1988

    Dentsply International — Marketing Organization

2020s

  1. Jan 1, 2020

    Earliest Phase 3 Sponsor(trial)

Indications

Mechanism of action

Combination products

  • carbocaine w/ neo-cobefrin

    with mepivacaine

    Also known as arestocaine hydrochloride w/ levonordefrin, isocaine hydrochloride w/ levonordefrin, polocaine w/ levonordefrin, scandonest l

  • ravocaine and novocain w/ neo-cobefrin

    with procaine merethoxylline, propoxycaine

Approval history

  • approvedSep 19, 1952

Chemistry & pharmacology

Loading structure…

SMILES

C[C@H](N)[C@H](O)C1=CC=C(O)C(O)=C1
Mol. weight
183.2044 g/mol

Oral

No

Parenteral

No

Topical

No

Sources

Clinical trials

NCT IDPhaseStart dateSponsor(s)
NCT05875519N/AMay 1, 2023Minia University
NCT04477317Phase 3Nov 30, 2020Cairo University
NCT04561921N/AOct 22, 2020Cairo University
Showing 3 of 3 trials
Page 1 / 1

Organizations

Research & Development (2)

OrganizationOrg typeTrialsAs lead sponsorPhasesEarliest year
Cairo UniversityAcademic/Hospital2222020
Minia UniversityAcademic/Hospital1112023
2 organizations
Page 1 / 1

Marketing (8)

OrganizationOrg typeRelationshipDate
BelmoraAcademic/HospitalMKTGJan 22, 1976
Dentsply InternationalFor profitMKTGApr 14, 1988
DeprocoFor profitMKTGOct 10, 1984
KodakFor profitNDA2Jan 6, 1960
KodakFor profitNDASep 19, 1952
SeptodontFor profitMKTGFeb 6, 1976
SeptodontFor profitSYNFeb 6, 1976
SolvayFor profitMKTGApr 15, 1976