← Mechanisms of action

Alpha-2 adrenergic receptor

PROTEIN FAMILYMus musculus

Linked proteins

Drugs acting on this target (5)

Active Pharmaceutical Ingredient Mechanism Type Approval Status API Type Mechanism of Action
lofexidine (lucemyra)ActivatorapprovedSmall moleculeAlpha-2 adrenergic receptor activator
levonordefrin (Neo-Cobefrine)AgonistapprovedSmall moleculeAlpha-2 adrenergic receptor agonist
medetomidineAgonistexperimentalSmall moleculeAlpha-2 adrenergic receptor agonist
oxymetazoline (ocuclear)AgonistapprovedSmall moleculeAlpha-2 adrenergic receptor agonist
atipamezole (Antisedan)AntagonistexperimentalSmall moleculeAlpha-2 adrenergic receptor antagonist