bezlotoxumab

Trade name: zinplava

mAbapprovedFast Track FDA

Approved

Oct 21, 2016

Bezlotoxumab, sold under the brand name Zinplava, is a human monoclonal antibody designed for the prevention of recurrence of Clostridioides difficile infections. Bezlotoxumab binds to Clostridioides difficile toxin B. — Wikipedia

Clinical trial activity

12 trials · 45 clinical orgs · 2 marketing orgs

Phase 1
0
Phase 2
6
Phase 3
3
Phase 4
6

Earliest trial started Jul 1, 2006 (NCT00350298)

Timeline

2000s

  1. Jan 1, 2006

    Earliest Phase 2 Sponsor(trial)

2010s

  1. Jan 1, 2011

    Merck — Earliest Phase 3 Sponsor(trial)

  2. Oct 21, 2016

    Merck — Earliest FDA Approval

  3. Oct 21, 2016

    Merck — Marketing Organization

  4. Oct 21, 2016

    Merck — NDA Organization

Indications

Mechanism of action

Approval history

  • approvedPriority reviewFast trackOct 21, 2016

Chemistry & pharmacology

Chirality
Single Stereoisomer
Inorganic
No
Polymer
No
Availability
Prescription Only
Multi-specific
No

Oral

No

Parenteral

No

Topical

No

First in class

Sources

Also known as

  • bezlotoxumab
  • bezlotoxumab
  • bezlotoxumab
  • bezlotoxumab
  • bezlotoxumab
  • bezlotoxumab
  • bezlotoxumab
  • bezlotoxumab
  • gs-cda1
  • gs-cda1
  • mdx-1388
  • mdx-1388
  • mk-6072
  • mk-6072
  • mk-6072
  • zinplava
  • zinplava

Clinical trials

NCT IDPhaseStart dateSponsor(s)
NCT05304715Phase 2Apr 13, 2022Hellenic Institute for the Study of Sepsis, Hellenic Sepsis Study Group
NCT05077085Phase 4Jan 31, 2022Erasmus University Rotterdam, Leiden University, Medical Center Haaglanden, OLVG hospital, Amsterdam, University of Amsterdam
NCT04626947Phase 4Nov 30, 2020Merck, University of Pittsburgh
NCT04415918Phase 4Jul 1, 2020Cooper Human Systems
NCT03937999Phase 4Jul 8, 2019Merck, Yeshiva University
NCT03880539Phase 4Jun 10, 2019Merck, University of Kansas
NCT03756454Phase 4Apr 30, 2019Merck, Ohio State University
NCT03829475Phase 2Mar 1, 2019Harvard University
NCT03182907Phase 3Dec 1, 2017Merck
NCT01513239Phase 3Feb 1, 2012Merck
NCT01241552Phase 3Oct 1, 2011Merck
NCT00350298Phase 2Jul 1, 2006Baylor University, Central Indiana Gastroenterology Group, Centre de Sante et de Services Sociaux de Chicoutimi, Centre Hospitalier Regional de Trois-Rivieres, Chest, Infectious Diseases and Critical Care Assoc., PC, Dr. Kiran C. Patel Research Institute, Henry Ford Health System, Icahn School of Medicine at Mount Sinai, Idaho Falls Infectious Diseases, PLLC, Jersey Shore University Medical Center, Kaiser Permanente, Mayo Clinic, Medarex, Mercury Street Medical Group, MultiCare Health System Research Institute, PMG Research, Queen's University, Belfast, Rapid City Regional Hospital, Remington-Davis Clinical Research, Saint Luke's Health System, Summa Health System, Texas A&M University, Thomas Jefferson University, University of Calgary, University of California, Los Angeles, University of Kentucky, University of Manitoba, University of Massachusetts, University of Southern California, Vancouver Island Health Research Centre, Windsor Regional Hospital
Showing 12 of 12 trials
Page 1 / 1

Organizations

Research & Development (45)

OrganizationOrg typeTrialsAs lead sponsorPhasesEarliest year
MerckFor profit7322011
Baylor UniversityAcademic/Hospital1012006
Central Indiana Gastroenterology GroupAcademic/Hospital1012006
Centre de Sante et de Services Sociaux de ChicoutimiAcademic/Hospital1012006
Centre Hospitalier Regional de Trois-RivieresAcademic/Hospital1012006
Chest, Infectious Diseases and Critical Care Assoc., PCAcademic/Hospital1012006
Cooper Human SystemsFor profit1112020
Dr. Kiran C. Patel Research InstituteAcademic/Hospital1012006
Erasmus University RotterdamAcademic/Hospital1012022
Harvard UniversityAcademic/Hospital1112019
Hellenic Institute for the Study of SepsisAcademic/Hospital1112022
Hellenic Sepsis Study GroupAcademic/Hospital1012022
Henry Ford Health SystemAcademic/Hospital1012006
Icahn School of Medicine at Mount SinaiAcademic/Hospital1012006
Idaho Falls Infectious Diseases, PLLCAcademic/Hospital1012006
Jersey Shore University Medical CenterAcademic/Hospital1012006
Kaiser PermanenteAcademic/Hospital1012006
Leiden UniversityAcademic/Hospital1112022
Mayo ClinicAcademic/Hospital1012006
MedarexFor profit1012006
45 organizations
Page 1 / 3

Marketing (3)

OrganizationOrg typeRelationshipDate
MedarexFor profitIND
MerckFor profitMKTGOct 21, 2016
MerckFor profitNDAOct 21, 2016