← Mechanisms of action

Soluble guanylate cyclase

PROTEIN COMPLEX GROUPHomo sapiens

Linked proteins

Drugs acting on this target (17)

Active Pharmaceutical Ingredient Mechanism Type Approval Status API Type Mechanism of Action
ataciguatActivatorexperimentalSmall moleculeactivator - GUCY1A2
cinaciguatActivatorexperimentalSmall moleculeSoluble guanylate cyclase activator
isosorbide (isordil)ActivatorapprovedSmall moleculeSoluble guanylate cyclase activator
iw-1973ActivatorexperimentalSmall moleculeactivator - GUCY1A2
nitric oxide (inomax)ActivatorapprovedSmall moleculeSoluble guanylate cyclase activator
nitroglycerin (transderm-nitro)ActivatorapprovedSmall moleculeSoluble guanylate cyclase activator
OlinciguatActivatorexperimentalSmall moleculeSoluble guanylate cyclase activator
praliciguatActivatorexperimentalSmall moleculeSoluble guanylate cyclase activator
runcaciguatActivatorexperimentalSmall moleculeSoluble guanylate cyclase activator
tetranitropentaerythritolActivatorexperimentalSmall moleculeSoluble guanylate cyclase activator
vericiguat (Verquvo)ActivatorapprovedSmall moleculeSoluble guanylate cyclase activator
iw-3300AgonistexperimentalSmall moleculeSoluble guanylate cyclase agonist
iw-9179AgonistexperimentalSmall moleculeSoluble guanylate cyclase agonist
vericiguat (Verquvo)AgonistapprovedSmall moleculeSoluble guanylate cyclase agonist
methylene blue (proveblue)InhibitorapprovedSmall moleculeSoluble guanylate cyclase inhibitor
OlinciguatPositive allosteric modulatorexperimentalSmall moleculeSoluble guanylate cyclase positive allosteric modulator
riociguat (adempas)Positive allosteric modulatorapprovedSmall moleculeSoluble guanylate cyclase positive allosteric modulator